SCHEMBL28645243

SCHEMBL28645243

COc1ccc([C@@H]2CNC(=O)[C@@H](c3ccc(F)cc3)C2)cc1OC

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 18/20 0.56
PDE4D Q08499 14/20 0.56
PDE4B Q07343 12/20 0.56
PDE4C Q08493 12/20 0.56
CYP3A4 P08684 2/20 0.46
VEGFA P15692 1/20 0.46
ALDH1A1 P00352 1/20 0.46
LMNA P02545 1/20 0.46
CYP1A2 P05177 1/20 0.46
MAPT P10636 1/20 0.46
CYP2C9 P11712 1/20 0.46
ALOX15 P16050 1/20 0.46
CREBBP Q92793 1/20 0.46
KDM4E B2RXH2 1/20 0.46
PDE5A O76074 1/20 0.46
TNF P01375 1/20 0.46
MAPK1 P28482 1/20 0.46
BLM P54132 1/20 0.46
PDE1A P54750 1/20 0.46
PDE1B Q01064 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30823798 1.00 PDE4A (0.56) PDE4APDE4DPDE4BPDE4CCYP3A4
SCHEMBL28645245 1.00 PDE4A (0.56) PDE4APDE4DPDE4BPDE4CCYP3A4
SCHEMBL28645237 0.83 FPR1 (0.48) ALDH1A1KDM4EKMT2A
SCHEMBL28645234 0.83 FPR1 (0.48) ALDH1A1KDM4EKMT2A
SCHEMBL28657641 0.79 HTR2C (0.41) PDE4DKMT2A
SCHEMBL28657639 0.79 HTR2C (0.41) PDE4DKMT2A
SCHEMBL28653227 0.77 MMP13 (0.40)
SCHEMBL28653229 0.77 MMP13 (0.40)
SCHEMBL2799305 0.76 PDE4A (0.57) PDE4APDE4DPDE4BPDE4C
SCHEMBL2799239 0.76 PDE4A (0.57) PDE4APDE4DPDE4BPDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113461599-B Process for preparing piperidone compounds 南方科技大学 2024-02-09 CN disclosed
CN-113461599-A Process for producing piperidone compound 南方科技大学 2021-10-01 CN disclosed