SCHEMBL28645604

SCHEMBL28645604

CC(C)n1cc(B2OC(C)(C)C(C)(C)O2)cc(F)c1=O

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LPL P06858 4/20 0.37
LIPG Q9Y5X9 4/20 0.37
ROCK1 Q13464 1/20 0.36
IDO1 P14902 1/20 0.34
TDO2 P48775 1/20 0.34
BACE1 P56817 3/20 0.32
F11 P03951 2/20 0.32
F2 P00734 1/20 0.32
PRSS1 P07477 1/20 0.32
PRSS2 P07478 1/20 0.32
PRSS3 P35030 1/20 0.32
FFAR1 O14842 1/20 0.31
CA1 P00915 3/20 0.31
CA2 P00918 3/20 0.31
CA9 Q16790 3/20 0.31
JAK2 O60674 2/20 0.31
BTK Q06187 2/20 0.31
CA12 O43570 1/20 0.31
CA3 P07451 1/20 0.31
CA4 P22748 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16650743 0.84 LPL (0.33) LPLLIPGIDO1TDO2BACE1
SCHEMBL22230214 0.82 AAK1 (0.34) LPLLIPGBACE1F11FFAR1
SCHEMBL22655363 0.81 LPL (0.36) LPLLIPGROCK1BACE1F11
SCHEMBL16650516 0.80 LPL (0.40) LPLLIPGROCK1IDO1TDO2
SCHEMBL22655301 0.80 CSF1R (0.38) LPLLIPGBACE1FFAR1CA1
SCHEMBL31752740 0.77 LPL (0.37) LPLLIPGROCK1IDO1TDO2
SCHEMBL505914 0.74 LPL (0.41) LPLLIPGBACE1F11FFAR1
SCHEMBL28647197 0.71 KDM4E (0.30)
SCHEMBL878145 0.70 F11 (0.34) LIPGBACE1F11F2PRSS1
SCHEMBL1106436 0.70 BRD4 (0.37)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109293652-B Substituted thiazole derivative and application thereof 四川科伦博泰生物医药股份有限公司 2021-10-22 CN disclosed