SCHEMBL28645763

SCHEMBL28645763

CCOc1cc2c(cc1C(=O)O)CN(CC(C)C)C2=O

nearest known ligand 0.48

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.41
PARP1 P09874 1/20 0.41
TSHR P16473 1/20 0.41
HSD17B10 Q99714 1/20 0.41
ALOX15 P16050 1/20 0.37
MEN1 O00255 1/20 0.36
NPC1 O15118 1/20 0.36
POLB P06746 1/20 0.36
PRMT5 O14744 1/20 0.35
WDR77 Q9BQA1 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28645772 0.88 PARP1 (0.40) KMT2APARP1MEN1NPC1POLB
SCHEMBL28645344 0.83 KMT2A (0.41) KMT2ATSHRHSD17B10ALOX15
SCHEMBL28633462 0.81 KMT2A (0.53) KMT2APARP1ALOX15MEN1
SCHEMBL28652352 0.80 KMT2A (0.48) KMT2APARP1TSHRALOX15
SCHEMBL28656930 0.79 KMT2A (0.45) KMT2ATSHRHSD17B10ALOX15MEN1
SCHEMBL30604606 0.79 KMT2A (0.45) KMT2ATSHRHSD17B10ALOX15MEN1
SCHEMBL30604612 0.79 KMT2A (0.47) KMT2ATSHRMEN1
SCHEMBL28638917 0.79 KMT2A (0.47) KMT2ATSHRMEN1
SCHEMBL28651754 0.76 KMT2A (0.49) KMT2ATSHRHSD17B10ALOX15MEN1
SCHEMBL30604611 0.76 ADAM17 (0.44) PARP1PRMT5WDR77

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113493438-B Tetrahydroisoquinoline compounds 南京再明医药有限公司 2023-10-20 CN disclosed
CN-113493438-A Tetrahydroisoquinoline compounds 江苏先声药业有限公司 2021-10-12 CN disclosed