SCHEMBL28645962

SCHEMBL28645962

CC(C)(C)OC(=O)NNC(=O)c1ccc(C(F)(F)F)nc1

nearest known ligand 0.56

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.43
POLB P06746 1/20 0.43
PTPN1 P18031 1/20 0.41
TRPV1 Q8NER1 1/20 0.39
SLC6A3 Q01959 1/20 0.39
KCNH2 Q12809 1/20 0.39
TAAR1 Q96RJ0 1/20 0.39
NAMPT P43490 1/20 0.38
SCN9A Q15858 1/20 0.38
APLNR P35414 1/20 0.38
MRGPRX4 Q96LA9 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30015957 1.00 LMNA (0.43) LMNAPOLBPTPN1TRPV1SLC6A3
SCHEMBL24599026 0.82 HDAC1 (0.55) LMNAPOLBNAMPT
SCHEMBL28632079 0.80 DDR1 (0.45) LMNAPOLB
SCHEMBL31512899 0.80 TRPV1 (0.50) LMNAPOLBTRPV1
SCHEMBL30850105 0.80 CA12 (0.48) PTPN1TRPV1SCN9AMRGPRX4
SCHEMBL15600325 0.80 GAA (0.43) LMNAPOLBTRPV1NAMPTSCN9A
SCHEMBL12322215 0.79 CA12 (0.40) LMNAPOLBPTPN1TRPV1NAMPT
SCHEMBL20581109 0.78 L3MBTL1 (0.51) LMNA
SCHEMBL20581110 0.78 L3MBTL1 (0.51) LMNA
SCHEMBL13701813 0.77 LMNA (0.46) LMNAPTPN1TRPV1SLC6A3KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113264945-B Spiro derivative, preparation method and medical application thereof 江苏恒瑞医药股份有限公司 2022-11-22 CN disclosed
CN-113264945-A Spiro derivative, preparation method and medical application thereof 江苏恒瑞医药股份有限公司 2021-08-17 CN disclosed