SCHEMBL28646100

SCHEMBL28646100

COC(=O)C(C)(C)N(CCCC(=O)O)Cc1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4A O75164 2/20 0.42
KDM4C Q9H3R0 2/20 0.42
HDAC3 O15379 2/20 0.41
HDAC1 Q13547 2/20 0.41
HDAC2 Q92769 2/20 0.41
HDAC8 Q9BY41 2/20 0.41
MAPK1 P28482 1/20 0.41
ADRA1A P35348 1/20 0.41
HDAC4 P56524 1/20 0.41
SLC6A3 Q01959 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
HDAC7 Q8WUI4 1/20 0.41
HDAC10 Q969S8 1/20 0.41
HDAC11 Q96DB2 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
HDAC9 Q9UKV0 1/20 0.41
HDAC5 Q9UQL6 1/20 0.41
HTT P42858 3/20 0.40
BMP1 P13497 1/20 0.40
LTA4H P09960 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21758682 0.91 LTA4H (0.46) HDAC3HDAC1HDAC2HDAC8HTT
SCHEMBL29151949 0.85 TDP1 (0.50) HTTLTA4HMEN1KMT2AL3MBTL1
SCHEMBL14350236 0.83 HTT (0.49) KDM4AKDM4CHDAC3HDAC1HDAC2
SCHEMBL14350197 0.79 KDM4A (0.50) KDM4AKDM4CHDAC3HDAC1HDAC2
SCHEMBL17540988 0.78 ALOX5 (0.54) MAPK1SMN1; SMN2HTTLTA4HMEN1
SCHEMBL14350209 0.77 KDM4A (0.52) KDM4AKDM4CHDAC3HDAC1HDAC2
SCHEMBL14350210 0.77 KDM4A (0.52) KDM4AKDM4CHDAC3HDAC1HDAC2
SCHEMBL14350200 0.77 KDM4A (0.52) KDM4AKDM4CHDAC3HDAC1HDAC2
SCHEMBL14350181 0.77 KDM4A (0.52) KDM4AKDM4CHDAC3HDAC1HDAC2
SCHEMBL14350189 0.76 KMT2A (0.51) KDM4AKDM4CHDAC3HDAC1HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112739698-A Tetrahydropyrimidine derivatives as AHR modulators 捷豹治疗有限公司 2021-04-30 CN disclosed