SCHEMBL28646266

SCHEMBL28646266

COc1cccc(C2=CC2(F)F)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 1/20 0.50
CLK4 Q9HAZ1 1/20 0.50
CYP3A4 P08684 2/20 0.48
CYP1A1 P04798 1/20 0.48
CYP1A2 P05177 1/20 0.48
CYP2E1 P05181 1/20 0.48
CYP2C8 P10632 1/20 0.48
CYP2D6 P10635 1/20 0.48
CYP2A6 P11509 1/20 0.48
CYP2C9 P11712 1/20 0.48
CYP4B1 P13584 1/20 0.48
CYP2B6 P20813 1/20 0.48
CYP3A5 P20815 1/20 0.48
CYP2A7 P20853 1/20 0.48
CYP3A7 P24462 1/20 0.48
CYP2F1 P24903 1/20 0.48
CYP2C18 P33260 1/20 0.48
CYP2C19 P33261 1/20 0.48
CYP2J2 P51589 1/20 0.48
CYP4F2 P78329 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29489425 0.79 CYP3A4 (0.73) DYRK1ACLK4CYP3A4CYP1A1CYP1A2
SCHEMBL196765 0.79 CYP3A4 (0.73) DYRK1ACLK4CYP3A4CYP1A1CYP1A2
SCHEMBL29628977 0.77 CYP3A4 (0.77) DYRK1ACLK4CYP3A4CYP1A1CYP1A2
Ammonia Solution, Strong SCHEMBL27960505 0.77 CYP3A4 (0.70) DYRK1ACLK4CYP3A4CYP1A1CYP1A2
Hydrogen Sulfide SCHEMBL28640169 0.77 CYP3A4 (0.70) DYRK1ACLK4CYP3A4CYP1A1CYP1A2
SCHEMBL28638395 0.75 CA1 (0.50) CLK4ACHEGAACA1CA2
SCHEMBL1180343 0.74 ABL1 (0.69) DYRK1ACLK4CYP3A4CYP1A1CYP1A2
SCHEMBL29279106 0.74 ACHE (0.46) CYP3A4CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL30753767 0.74 ACHE (0.46) CYP3A4CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL5620245 0.73 CYP3A4 (0.86) DYRK1ACLK4CYP3A4CYP1A1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113480476-B 4-fluoropyridine derivative and preparation method and application thereof 山东师范大学 2022-07-22 CN claimed
CN-113480476-A 4-fluoropyridine derivative and preparation method and application thereof 山东师范大学 2021-10-08 CN claimed
CN-113480476-B 4-fluoropyridine derivative and preparation method and application thereof 山东师范大学 2022-07-22 CN disclosed
CN-113480476-A 4-fluoropyridine derivative and preparation method and application thereof 山东师范大学 2021-10-08 CN disclosed