SCHEMBL28647880

SCHEMBL28647880

CC(C)(C)OC(=O)N1CCCC(c2cn(-c3ccc(OCc4ccccn4)c(Cl)c3)c3c(N)ncnc23)C1

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
EGFR P00533 13/20 0.45
ERBB2 P04626 11/20 0.45
BTK Q06187 2/20 0.45
BLK P51451 1/20 0.45
BMX P51813 1/20 0.45
MAP2K1 Q02750 1/20 0.45
ERBB4 Q15303 1/20 0.45
KDM1A O60341 1/20 0.37
SRC P12931 2/20 0.37
AURKA O14965 1/20 0.36
RPS6KB1 P23443 1/20 0.36
ABL1 P00519 1/20 0.36
ABL2 P42684 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28859066 0.88 BTK (0.58) EGFRERBB2BTKBLKBMX
SCHEMBL29989719 0.87 BTK (0.46) EGFRERBB2BTKBLKBMX
SCHEMBL28645870 0.87 BTK (0.46) EGFRERBB2BTKBLKBMX
SCHEMBL28925175 0.85 KDM1A (0.43) EGFRERBB2BTKBLKBMX
SCHEMBL29989219 0.80 SLC6A4 (0.40) EGFRERBB2BTKBLKBMX
SCHEMBL28645873 0.80 SLC6A4 (0.40) EGFRERBB2BTKBLKBMX
SCHEMBL28636590 0.80 KDM1A (0.38) EGFRERBB2BTKBLKBMX
SCHEMBL29989351 0.79 BTK (0.48) EGFRERBB2BTKBLKBMX
SCHEMBL21044817 0.79 BTK (0.53) BTK
SCHEMBL28636595 0.78 BTK (0.45) EGFRERBB2BTKBLKBMX

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113493439-B Substituted acrylamide derivative, composition and application thereof 深圳市塔吉瑞生物医药有限公司 2022-10-14 CN disclosed
CN-113493439-A Substituted acrylamide derivative, composition and application thereof 深圳市塔吉瑞生物医药有限公司 2021-10-12 CN disclosed