SCHEMBL28645873

SCHEMBL28645873

Nc1ncnc2c(C3CCCNC3)cn(-c3ccc(OCc4ccccn4)c(Cl)c3)c12

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 1/20 0.40
ERBB2 P04626 12/20 0.38
EGFR P00533 11/20 0.38
BTK Q06187 3/20 0.38
ERBB4 Q15303 2/20 0.38
MAP4K3 Q8IVH8 1/20 0.38
BLK P51451 1/20 0.38
BMX P51813 1/20 0.38
MAP2K1 Q02750 1/20 0.38
IGF1R P08069 1/20 0.36
SYK P43405 1/20 0.36
AURKA O14965 1/20 0.36
RPS6KB1 P23443 1/20 0.36
ERBB3 P21860 1/20 0.36
HTR2A P28223 1/20 0.36
HTR2C P28335 1/20 0.36
KCNH2 Q12809 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29989219 1.00 SLC6A4 (0.40) SLC6A4ERBB2EGFRBTKERBB4
SCHEMBL28956018 0.85 BTK (0.47) SLC6A4ERBB2EGFRBTKERBB4
SCHEMBL29989278 0.85 BTK (0.47) SLC6A4ERBB2EGFRBTKERBB4
SCHEMBL28859066 0.81 BTK (0.58) ERBB2EGFRBTKERBB4BLK
SCHEMBL28647880 0.80 EGFR (0.45) ERBB2EGFRBTKERBB4BLK
SCHEMBL8819946 0.78 BTK (0.43) SLC6A4EGFRBTKKCNH2
SCHEMBL29989239 0.76 ACVRL1 (0.54) SLC6A4ERBB2EGFRBTKERBB4
SCHEMBL19230428 0.76 BTK (0.56) BTK
SCHEMBL29989357 0.75 TNK2 (0.53) ERBB2EGFRBTKERBB4BLK
SCHEMBL409545 0.74 HTR6 (0.43) EGFRBTKRPS6KB1HTR2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113493439-B Substituted acrylamide derivative, composition and application thereof 深圳市塔吉瑞生物医药有限公司 2022-10-14 CN disclosed
CN-113493439-A Substituted acrylamide derivative, composition and application thereof 深圳市塔吉瑞生物医药有限公司 2021-10-12 CN disclosed