SCHEMBL28648019

SCHEMBL28648019

CC1C=CC(NC(=O)OC(C)(C)C)=CN1C(=O)O

nearest known ligand 0.38

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NFKB1 P19838 6/20 0.38
NFKB2 Q00653 6/20 0.38
RELA Q04206 6/20 0.38
MAPT P10636 1/20 0.32
BCL2 P10415 2/20 0.32
CYP17A1 P05093 1/20 0.32
NAMPT P43490 1/20 0.32
BECN1 Q14457 1/20 0.31
IDO1 P14902 1/20 0.31
BRD9 Q9H8M2 1/20 0.31
KDM4E B2RXH2 1/20 0.30
PKM P14618 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31258505 0.68 NFKB1 (0.35) NFKB1NFKB2RELACYP17A1
SCHEMBL18901801 0.67 NFKB1 (0.40) NFKB1NFKB2RELACYP17A1
SCHEMBL18929421 0.65 NFKB1 (0.38) NFKB1NFKB2RELACYP17A1
SCHEMBL29893827 0.64 NFKB1 (0.40) NFKB1NFKB2RELAMAPTCYP17A1
SCHEMBL14138294 0.63 NFKB1 (0.35) NFKB1NFKB2RELA
SCHEMBL19056136 0.62 NFKB1 (0.39) NFKB1NFKB2RELA
SCHEMBL27991298 0.61 NFKB1 (0.42) NFKB1NFKB2RELACYP17A1
SCHEMBL28269645 0.61 NFKB1 (0.42) NFKB1NFKB2RELACYP17A1
SCHEMBL19512667 0.61 NFKB1 (0.40) NFKB1NFKB2RELACYP17A1NAMPT
SCHEMBL13055402 0.60 CYP17A1 (0.59) CYP17A1NAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113677346-A Inhibitors of cyclin dependent kinase 7(CDK7) 希洛斯医药品股份有限公司 2021-11-19 CN disclosed
CN-113226306-A Methods of treating cancer in a patient identified by a biomarker using a non-covalent inhibitor of cyclin dependent kinase 7(CDK7) 希洛斯医药品股份有限公司 2021-08-06 CN disclosed