SCHEMBL18901801

SCHEMBL18901801

COC(=O)C1C=CC(NC(=O)OC(C)(C)C)=C1

nearest known ligand 0.40

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
NFKB1 P19838 7/20 0.40
NFKB2 Q00653 7/20 0.40
RELA Q04206 7/20 0.40
ATR Q13535 1/20 0.37
ALDH1A1 P00352 1/20 0.34
GAA P10253 1/20 0.34
CYP17A1 P05093 1/20 0.32
PTGDR2 Q9Y5Y4 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18929421 0.77 NFKB1 (0.38) NFKB1NFKB2RELAATRALDH1A1
SCHEMBL14138294 0.69 NFKB1 (0.35) NFKB1NFKB2RELAATRALDH1A1
SCHEMBL19056136 0.68 NFKB1 (0.39) NFKB1NFKB2RELAATR
SCHEMBL31258505 0.68 NFKB1 (0.35) NFKB1NFKB2RELAATRCYP17A1
SCHEMBL20224875 0.67 MAPK1 (0.39) NFKB1NFKB2RELA
SCHEMBL28648019 0.67 NFKB1 (0.38) NFKB1NFKB2RELACYP17A1
SCHEMBL29893827 0.67 NFKB1 (0.40) NFKB1NFKB2RELAATRGAA
SCHEMBL19512667 0.64 NFKB1 (0.40) NFKB1NFKB2RELAATRALDH1A1
SCHEMBL11076557 0.63 DNTT (0.37) ALDH1A1
SCHEMBL13055402 0.63 CYP17A1 (0.59) ALDH1A1GAACYP17A1PTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1763351-B9 3-AMINOCYCLOPENTANECARBOXAMIDES AS MODULATORS OF CHEMOKINE RECEPTORS INCYTE HOLDINGS CORP (US) 2017-05-31 EP disclosed