SCHEMBL28649130

SCHEMBL28649130

COC(=O)c1cc(-n2cnc(C3CC3)c2)ccc1C

nearest known ligand 0.45

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 1/20 0.45
GRM1 Q13255 1/20 0.45
MAP3K5 Q99683 16/20 0.44
RIPK2 O43353 2/20 0.40
KDM4E B2RXH2 1/20 0.39
MAPT P10636 1/20 0.39
ALOX15 P16050 1/20 0.39
TSHR P16473 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28648560 0.87 GRM5 (0.44) GRM5GRM1MAP3K5MAPT
SCHEMBL28663394 0.87 MAP3K5 (0.46) GRM5GRM1MAP3K5RIPK2TSHR
SCHEMBL28648131 0.86 MAP3K5 (0.44) MAP3K5RIPK2
SCHEMBL28660344 0.85 MAP3K5 (0.43) MAP3K5RIPK2
SCHEMBL20672216 0.80 MAP3K5 (0.43) GRM5GRM1MAP3K5RIPK2ALOX15
SCHEMBL30028786 0.80 MAP3K5 (0.43) GRM5GRM1MAP3K5RIPK2ALOX15
SCHEMBL28643803 0.80 MAP3K5 (0.53) GRM5GRM1MAP3K5MAPT
SCHEMBL21461103 0.80 MAP3K5 (0.52) GRM5GRM1MAP3K5
SCHEMBL28656996 0.79 MAP3K5 (0.53) GRM5GRM1MAP3K5RIPK2
SCHEMBL234409 0.79 MAP3K5 (0.43) GRM5GRM1MAP3K5MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109400625-B Fused bicyclic compound and application thereof in medicine 广东东阳光药业有限公司 2021-11-12 CN disclosed