SCHEMBL30028786

SCHEMBL30028786

COC(=O)c1ccc2cc(-n3cnc(C4CC4)c3)ccc2c1

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MAP3K5 Q99683 10/20 0.43
GRM5 P41594 1/20 0.40
GRM1 Q13255 1/20 0.40
HTT P42858 2/20 0.40
ALOX15 P16050 1/20 0.40
PTPN11 Q06124 1/20 0.40
RIPK2 O43353 2/20 0.39
CYP19A1 P11511 1/20 0.39
CYP11B1 P15538 1/20 0.39
CYP11B2 P19099 1/20 0.39
FGFR1 P11362 1/20 0.38
ALDH1A1 P00352 1/20 0.38
ATM Q13315 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20672216 1.00 MAP3K5 (0.43) MAP3K5GRM5GRM1HTTALOX15
SCHEMBL28643803 0.86 MAP3K5 (0.53) MAP3K5GRM5GRM1FGFR1ALDH1A1
SCHEMBL30029659 0.85 MAP3K5 (0.42) MAP3K5RIPK2
SCHEMBL20672223 0.85 MAP3K5 (0.42) MAP3K5RIPK2
SCHEMBL28656996 0.80 MAP3K5 (0.53) MAP3K5GRM5GRM1RIPK2ALDH1A1
SCHEMBL28649130 0.80 GRM5 (0.45) MAP3K5GRM5GRM1ALOX15RIPK2
SCHEMBL28658681 0.80 TLR2 (0.44) MAP3K5GRM5GRM1RIPK2ALDH1A1
SCHEMBL28654034 0.79 MAP3K5 (0.48) MAP3K5GRM5GRM1
SCHEMBL28648560 0.79 GRM5 (0.44) MAP3K5GRM5GRM1FGFR1
SCHEMBL28649133 0.79 MAP3K5 (0.44) MAP3K5GRM5GRM1ALDH1A1ATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109265443-B Heterocyclic compounds as ASK inhibitors and uses thereof 南京圣和药业股份有限公司 2022-11-29 CN disclosed