SCHEMBL28656996

SCHEMBL28656996

COC(=O)c1ccc(C)c(-n2cnc(C3CC3)c2)c1

nearest known ligand 0.53

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MAP3K5 Q99683 15/20 0.53
TLR2 O60603 1/20 0.44
TLR1 Q15399 1/20 0.44
RIPK2 O43353 1/20 0.43
ALDH1A1 P00352 1/20 0.43
GRM5 P41594 1/20 0.41
GRM1 Q13255 1/20 0.41
ABL1 P00519 1/20 0.41
MAP3K6 O95382 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28658681 0.88 TLR2 (0.44) MAP3K5TLR2TLR1RIPK2ALDH1A1
SCHEMBL28649133 0.87 MAP3K5 (0.44) MAP3K5TLR2TLR1ALDH1A1GRM5
SCHEMBL28654034 0.87 MAP3K5 (0.48) MAP3K5TLR2TLR1GRM5GRM1
SCHEMBL28649418 0.86 MAP3K5 (0.53) MAP3K5RIPK2
SCHEMBL28643374 0.85 MAP3K5 (0.52) MAP3K5
SCHEMBL28643394 0.81 ALDH1A1 (0.41) MAP3K5ALDH1A1
SCHEMBL30028786 0.80 MAP3K5 (0.43) MAP3K5RIPK2ALDH1A1GRM5GRM1
SCHEMBL20672216 0.80 MAP3K5 (0.43) MAP3K5RIPK2ALDH1A1GRM5GRM1
SCHEMBL20802811 0.80 MAP3K5 (0.52) MAP3K5MAP3K6
SCHEMBL28646401 0.80 KDM4C (0.46) MAP3K5GRM5GRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109400625-B Fused bicyclic compound and application thereof in medicine 广东东阳光药业有限公司 2021-11-12 CN disclosed