SCHEMBL28649665

SCHEMBL28649665

COc1ncc(Br)cc1C(C)C

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 1/20 0.41
GABRB1 P18505 1/20 0.41
P2RX3 P56373 8/20 0.35
P2RX2 Q9UBL9 8/20 0.35
PIK3CA P42336 2/20 0.33
POLB P06746 1/20 0.33
GAA P10253 1/20 0.33
GFER P55789 1/20 0.33
MTOR P42345 1/20 0.33
PIK3R1 P27986 1/20 0.33
DYRK1B Q9Y463 2/20 0.33
HTT P42858 1/20 0.32
KMT2A Q03164 1/20 0.32
RORC P51449 1/20 0.32
MAPT P10636 1/20 0.32
CASP1 P29466 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29527168 1.00 GABRA1 (0.41) GABRA1GABRB1P2RX3P2RX2PIK3CA
SCHEMBL9948731 0.83 PIK3CA (0.33) PIK3CAMTORDYRK1BHTTKMT2A
SCHEMBL5781035 0.83 PIK3CA (0.33) PIK3CAMTORDYRK1BHTTKMT2A
SCHEMBL18751309 0.83 GABRA1 (0.39) GABRA1GABRB1HTTKMT2A
SCHEMBL15314666 0.79 GABRA1 (0.30) GABRA1GABRB1
SCHEMBL16133709 0.78 GABRA1 (0.35) GABRA1P2RX3P2RX2PIK3CAMTOR
SCHEMBL15292546 0.78 PIK3R1 (0.36) P2RX3P2RX2PIK3CAPOLBGAA
SCHEMBL31451331 0.78 TSHR (0.34) PIK3CAGAAMTORMAPT
SCHEMBL22959247 0.77 PIK3R1 (0.35) GABRA1GABRB1P2RX3P2RX2PIK3CA
SCHEMBL11890406 0.77 TSHR (0.43) GABRA1GABRB1P2RX3P2RX2PIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113698388-B 6-oxo-1, 6-dihydropyridine derivative, preparation method and application thereof in medicine 江苏恒瑞医药股份有限公司 2022-11-22 CN disclosed
CN-113698388-A 6-oxo-1, 6-dihydropyridine derivatives, preparation method and application thereof in medicines 江苏恒瑞医药股份有限公司 2021-11-26 CN disclosed