SCHEMBL28652009

SCHEMBL28652009

COc1ccc(-n2cnc(C3CC3)c2)cc1C(N)=O

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MAP3K5 Q99683 7/20 0.43
MAPT P10636 4/20 0.41
ACVR1 Q04771 1/20 0.39
TP53 P04637 1/20 0.38
SIK1 P57059 1/20 0.38
SIK2 Q9H0K1 1/20 0.38
SIK3 Q9Y2K2 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
ABL1 P00519 1/20 0.38
SYK P43405 1/20 0.37
PDE4A P27815 1/20 0.37
PDE4B Q07343 1/20 0.37
PDE4C Q08493 1/20 0.37
PDE4D Q08499 1/20 0.37
PARP15 Q460N3 1/20 0.37
PARP10 Q53GL7 1/20 0.37
GRM5 P41594 1/20 0.36
GRM1 Q13255 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL234409 0.89 MAP3K5 (0.43) MAP3K5MAPTABL1GRM5GRM1
SCHEMBL28648560 0.88 GRM5 (0.44) MAP3K5MAPTTP53KMT2AABL1
SCHEMBL28643811 0.88 MAP3K5 (0.43) MAP3K5MAPTTP53ABL1GRM5
SCHEMBL233653 0.84 MAP3K5 (0.44) MAP3K5MAPTABL1
SCHEMBL28643381 0.79 MAPK1 (0.43) MAP3K5ABL1PDE4APDE4BPDE4C
SCHEMBL28649130 0.78 GRM5 (0.45) MAP3K5MAPTGRM5GRM1
SCHEMBL28538145 0.77 MAP3K5 (0.41) MAP3K5GRM5GRM1
SCHEMBL28663394 0.77 MAP3K5 (0.46) MAP3K5GRM5GRM1
SCHEMBL28648131 0.76 MAP3K5 (0.44) MAP3K5
SCHEMBL28663432 0.75 MAP3K5 (0.41) MAP3K5PDE4APDE4BPDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109400625-B Fused bicyclic compound and application thereof in medicine 广东东阳光药业有限公司 2021-11-12 CN disclosed