SCHEMBL28652113

SCHEMBL28652113

COc1ccc(-c2ccccc2)cc1S(=O)(=O)Nc1ccc(C(=O)O)c(O)c1

nearest known ligand 0.64

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ACLY P53396 5/20 0.64
ALPL P05186 1/20 0.58
TRIM24 O15164 1/20 0.58
WDR5 P61964 1/20 0.56
ALDH1A1 P00352 2/20 0.56
HSD17B10 Q99714 2/20 0.56
PFKFB3 Q16875 1/20 0.56
MEN1 O00255 2/20 0.54
KMT2A Q03164 2/20 0.54
HPGD P15428 2/20 0.54
USP2 O75604 2/20 0.54
TSHR P16473 1/20 0.54
MCL1 Q07820 2/20 0.53
FABP4 P15090 1/20 0.53
GAA P10253 1/20 0.51
HCRTR2 O43614 1/20 0.51
TDP1 Q9NUW8 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28637913 0.91 ACLY (0.63) ACLYALPLTRIM24WDR5ALDH1A1
SCHEMBL28657533 0.91 ACLY (0.53) ACLYALPLTRIM24WDR5ALDH1A1
SCHEMBL28644506 0.88 ALDH1A1 (0.53) ACLYALPLTRIM24ALDH1A1HSD17B10
SCHEMBL28639303 0.88 MCL1 (0.64) ACLYALDH1A1HSD17B10PFKFB3MEN1
SCHEMBL9997390 0.87 PFKFB3 (0.65) ACLYTRIM24ALDH1A1HSD17B10PFKFB3
SCHEMBL28651873 0.86 PFKFB3 (0.53) ACLYALPLTRIM24ALDH1A1HSD17B10
SCHEMBL28637321 0.86 PFKFB3 (0.62) ACLYALDH1A1HSD17B10PFKFB3MEN1
SCHEMBL28647932 0.85 ALDH1A1 (0.70) ACLYALDH1A1HSD17B10PFKFB3MEN1
SCHEMBL28637063 0.84 ALDH1A1 (0.58) ACLYALDH1A1HSD17B10PFKFB3MEN1
SCHEMBL28639860 0.84 ALDH1A1 (0.53) ACLYALDH1A1HSD17B10PFKFB3MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113396145-A PFKFB3 inhibitors and uses thereof 盖罗发现有限责任公司 2021-09-14 CN disclosed