SCHEMBL28653236

SCHEMBL28653236

COc1cc(C(=O)Nc2ccc(N)cc2)cc(OC)c1OC

nearest known ligand 0.74

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 1/20 0.74
LMNA P02545 6/20 0.70
MAPT P10636 5/20 0.70
MEN1 O00255 4/20 0.70
KMT2A Q03164 4/20 0.70
ALDH1A1 P00352 2/20 0.70
MCL1 Q07820 2/20 0.70
MAPK1 P28482 1/20 0.70
GFER P55789 1/20 0.70
SMN1; SMN2 Q16637 2/20 0.68
TP53 P04637 1/20 0.68
GAA P10253 3/20 0.63
KDM4E B2RXH2 1/20 0.63
ABCG2 Q9UNQ0 1/20 0.61
POLB P06746 2/20 0.60
PKM P14618 1/20 0.57
APEX1 P27695 1/20 0.57
TDP1 Q9NUW8 1/20 0.57
SNCA P37840 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12584908 0.86 ABCB1 (0.76) ABCB1LMNAMAPTMEN1KMT2A
SCHEMBL9190681 0.86 ABCB1 (0.76) ABCB1LMNAMAPTMEN1KMT2A
SCHEMBL21409745 0.86 MEN1 (0.59) ABCB1LMNAMAPTMEN1KMT2A
Hydrochloric Acid SCHEMBL3718293 0.85 ALDH1A1 (0.69) ABCB1LMNAMAPTMEN1KMT2A
SCHEMBL1458219 0.85 ABCB1 (0.74) ABCB1LMNAMAPTMEN1KMT2A
SCHEMBL16656727 0.85 ABCB1 (0.74) ABCB1LMNAMAPTMEN1KMT2A
SCHEMBL1458094 0.85 MEN1 (0.74) ABCB1LMNAMAPTMEN1KMT2A
SCHEMBL707585 0.84 MEN1 (0.89) ABCB1LMNAMAPTMEN1KMT2A
SCHEMBL5148402 0.84 MEN1 (0.60) ABCB1LMNAMAPTMEN1KMT2A
SCHEMBL28707478 0.84 AURKB (0.67) ABCB1LMNAMEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113549043-B Flavonoid tankyrase 2 inhibitor and preparation method and application thereof 上海应用技术大学 2022-10-14 CN disclosed
CN-113461612-B Quinolone tankyrase 2 inhibitor and preparation method and application thereof 上海应用技术大学 2022-10-14 CN disclosed
CN-113549043-A Flavonoid tankyrase 2 inhibitor and preparation method and application thereof 上海应用技术大学 2021-10-26 CN disclosed
CN-113461612-A Quinolone tankyrase 2 inhibitor and preparation method and application thereof 上海应用技术大学 2021-10-01 CN disclosed