SCHEMBL28654034

SCHEMBL28654034

COC(=O)c1ccc(F)c(-n2cnc(C3CC3)c2)c1

nearest known ligand 0.48

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MAP3K5 Q99683 15/20 0.48
TLR2 O60603 1/20 0.45
TLR1 Q15399 1/20 0.45
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
ABL1 P00519 1/20 0.42
GRM5 P41594 1/20 0.40
GRM1 Q13255 1/20 0.40
MAP3K6 O95382 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28658681 0.87 TLR2 (0.44) MAP3K5TLR2TLR1CYP1A2CYP2C19
SCHEMBL28656996 0.87 MAP3K5 (0.53) MAP3K5TLR2TLR1ABL1GRM5
SCHEMBL28649133 0.86 MAP3K5 (0.44) MAP3K5TLR2TLR1ABL1GRM5
SCHEMBL28848812 0.81 MAP3K5 (0.51) MAP3K5
SCHEMBL28663394 0.79 MAP3K5 (0.46) MAP3K5GRM5GRM1MAP3K6
SCHEMBL20672216 0.79 MAP3K5 (0.43) MAP3K5GRM5GRM1
SCHEMBL30028786 0.79 MAP3K5 (0.43) MAP3K5GRM5GRM1
SCHEMBL28643803 0.79 MAP3K5 (0.53) MAP3K5CYP1A2CYP2C19GRM5GRM1
SCHEMBL28646401 0.79 KDM4C (0.46) MAP3K5GRM5GRM1
SCHEMBL19258658 0.78 MAP3K5 (0.64) MAP3K5MAP3K6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109400625-B Fused bicyclic compound and application thereof in medicine 广东东阳光药业有限公司 2021-11-12 CN disclosed