SCHEMBL28654591

SCHEMBL28654591

COc1cc(CNc2ccccn2)ccc1OCc1ccccc1Cl

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 5/20 0.70
KMT2A Q03164 5/20 0.70
SMN1; SMN2 Q16637 3/20 0.70
LMNA P02545 2/20 0.70
GAA P10253 2/20 0.60
L3MBTL1 Q9Y468 4/20 0.58
CYP1A2 P05177 2/20 0.58
CYP3A4 P08684 2/20 0.58
CYP2D6 P10635 2/20 0.58
CYP2C19 P33261 2/20 0.58
HTT P42858 1/20 0.56
CYP2C9 P11712 1/20 0.53
TP53 P04637 1/20 0.53
RAB9A P51151 2/20 0.52
NPC1 O15118 1/20 0.52
NFKB1 P19838 1/20 0.52
NFKB2 Q00653 1/20 0.52
RELA Q04206 1/20 0.52
SMARCA2 P51531 1/20 0.51
KDM4E B2RXH2 2/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28671557 0.90 MEN1 (0.72) MEN1KMT2ASMN1; SMN2LMNAGAA
SCHEMBL28653579 0.90 KMT2A (0.56) MEN1KMT2ASMN1; SMN2LMNAGAA
SCHEMBL28669019 0.89 MEN1 (0.57) MEN1KMT2ASMN1; SMN2LMNAGAA
SCHEMBL28654555 0.88 RAB9A (0.66) MEN1KMT2ASMN1; SMN2LMNAGAA
SCHEMBL28657460 0.87 GAA (0.60) MEN1KMT2ASMN1; SMN2LMNAGAA
SCHEMBL28659168 0.85 LMNA (0.61) MEN1KMT2ASMN1; SMN2LMNAGAA
SCHEMBL1633208 0.84 CXCR4 (0.63) MEN1KMT2ASMN1; SMN2LMNAGAA
SCHEMBL28659351 0.84 MEN1 (0.51) MEN1KMT2ASMN1; SMN2LMNAGAA
SCHEMBL28651416 0.83 SMARCA2 (0.72) MEN1KMT2ASMN1; SMN2LMNAGAA
SCHEMBL28654462 0.83 TP53 (0.55) MEN1KMT2ASMN1; SMN2LMNAGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109651365-B 3-methylpyrido [1,2-a ] pyrimidone derivative containing 1- ((4-substituted benzyl) oxy) and application thereof 贵州大学 2021-11-16 CN disclosed