SCHEMBL2865542

SCHEMBL2865542

O=C(CC(=O)OCC(=O)c1ccc(C(F)(F)F)cc1)OCC(=O)c1ccc(C(F)(F)F)cc1

nearest known ligand 0.70

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.70
MAPT P10636 1/20 0.70
PTPN1 P18031 2/20 0.56
GSK3B P49841 1/20 0.56
MMP1 P03956 1/20 0.53
CES2 O00748 1/20 0.50
CES1 P23141 1/20 0.50
HDAC1 Q13547 1/20 0.49
HDAC8 Q9BY41 1/20 0.49
MMP2 P08253 1/20 0.48
MMP8 P22894 1/20 0.48
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
GRM4 Q14833 1/20 0.47
HSD11B1 P28845 1/20 0.45
SRD5A2 P31213 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2865544 0.92 MAPT (0.65) ALDH1A1MAPTPTPN1GSK3BMMP1
SCHEMBL2749609 0.81 ALDH1A1 (0.60) ALDH1A1MAPTPTPN1GSK3BMMP1
SCHEMBL18329404 0.80 ALDH1A1 (0.59) ALDH1A1MAPTPTPN1GSK3BMMP1
SCHEMBL20355706 0.80 ALDH1A1 (0.55) ALDH1A1MAPTPTPN1GSK3BMMP1
SCHEMBL1349394 0.80 PTPN1 (0.57) ALDH1A1MAPTPTPN1GSK3BMMP1
SCHEMBL11686883 0.79 MAPT (0.58) ALDH1A1MAPTPTPN1GSK3BMMP1
SCHEMBL29987081 0.79 PTPN1 (0.75) ALDH1A1MAPTPTPN1GSK3BMMP1
SCHEMBL13731810 0.79 ALDH1A1 (0.61) ALDH1A1MAPTPTPN1GSK3BMMP1
SCHEMBL13731809 0.79 ALDH1A1 (0.61) ALDH1A1MAPTPTPN1GSK3BMMP1
SCHEMBL3391803 0.79 ALDH1A1 (0.60) ALDH1A1MAPTPTPN1GSK3BMMP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1805141-B1 PIPERIDINES AND RELATED COMPOUNDS FOR TREATMENT OF ALZHEIMER'S DISEASE MERCK SHARP & DOHME (GB) 2010-01-20 EP disclosed