SCHEMBL28655554

SCHEMBL28655554

CC(C)(C)c1ccc(C(=O)NC(=O)Nc2ccc(NC(=O)c3ccccc3)cc2)cc1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNK9 Q9NPC2 1/20 0.67
NPC1 O15118 3/20 0.66
RAB9A P51151 3/20 0.66
MEN1 O00255 1/20 0.66
KMT2A Q03164 1/20 0.66
NR1H4 Q96RI1 3/20 0.63
HDAC3 O15379 1/20 0.63
HDAC11 Q96DB2 1/20 0.63
HDAC8 Q9BY41 1/20 0.63
HDAC6 Q9UBN7 1/20 0.63
EPHX2 P34913 1/20 0.63
TRPV1 Q8NER1 4/20 0.61
SMN1; SMN2 Q16637 1/20 0.61
SIRT1 Q96EB6 2/20 0.61
CACNA1B Q00975 1/20 0.58
APBA1 Q02410 1/20 0.58
TP53 P04637 1/20 0.58
KDM4E B2RXH2 1/20 0.57
POLB P06746 1/20 0.57
CTDSP1 Q9GZU7 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19501539 0.89 NR1H4 (0.73) KCNK9NPC1RAB9AMEN1KMT2A
SCHEMBL7302565 0.89 KCNK9 (0.76) KCNK9NPC1RAB9AMEN1KMT2A
SCHEMBL4250752 0.86 KCNK9 (0.81) KCNK9NPC1RAB9ANR1H4HDAC3
SCHEMBL2345780 0.86 EPHX1 (0.68) KCNK9NPC1RAB9AMEN1KMT2A
SCHEMBL8218803 0.85 NR1H4 (0.63) NPC1RAB9AMEN1KMT2ANR1H4
SCHEMBL7303163 0.84 HDAC3 (0.86) NPC1RAB9AMEN1KMT2ANR1H4
SCHEMBL3404122 0.84 NR1H4 (0.60) NPC1RAB9AMEN1KMT2ANR1H4
SCHEMBL907217 0.84 EPHX2 (0.60) NPC1RAB9AMEN1KMT2ANR1H4
SCHEMBL12044572 0.83 PTPN1 (0.70) KCNK9NPC1RAB9ANR1H4HDAC3
SCHEMBL30994891 0.83 KCNK9 (0.72) KCNK9NPC1RAB9AMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113582969-A Application of acylthiourea compound in preparation of anti-enterovirus drugs 武汉大学 2021-11-02 CN claimed