SCHEMBL28657359

SCHEMBL28657359

Sc1ccccc1-c1cc2ccccc2c2ccccc12

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.50
HSD17B10 Q99714 4/20 0.50
HIF1A Q16665 3/20 0.50
TSHR P16473 3/20 0.50
HPGD P15428 2/20 0.50
MAPK1 P28482 2/20 0.50
CASP1 P29466 2/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
TRPM4 Q8TD43 1/20 0.45
CYP1B1 Q16678 1/20 0.44
CYP11B1 P15538 1/20 0.43
HPRT1 P00492 3/20 0.42
NISCH Q9Y2I1 1/20 0.41
CYP2A6 P11509 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
POLB P06746 1/20 0.37
MAPT P10636 1/20 0.37
PKM P14618 1/20 0.37
RAD52 P43351 1/20 0.37
TAAR1 Q96RJ0 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29637136 0.83 ALDH1A1 (0.60) ALDH1A1HSD17B10HIF1ATSHRHPGD
SCHEMBL7905250 0.83 ALDH1A1 (0.60) ALDH1A1HSD17B10HIF1ATSHRHPGD
SCHEMBL28654498 0.80 CYP2A6 (0.38) ALDH1A1HSD17B10HIF1ATSHRHPGD
SCHEMBL4442152 0.79 ALDH1A1 (0.55) ALDH1A1HSD17B10HIF1ATSHRHPGD
SCHEMBL28224726 0.78 CES1 (0.47) ALDH1A1HSD17B10HIF1ATSHRHPGD
SCHEMBL1436826 0.77 PTPN1 (0.46) ALDH1A1HSD17B10TSHRHPGDHPRT1
SCHEMBL28067095 0.77 ALDH1A1 (0.59) ALDH1A1HSD17B10HIF1ATSHRHPGD
SCHEMBL27520658 0.77 ALDH1A1 (0.40) ALDH1A1HSD17B10HIF1ATSHRHPGD
SCHEMBL4308375 0.77 ALDH1A1 (0.52) ALDH1A1HSD17B10HIF1ATSHRHPGD
SCHEMBL28968712 0.76 HPRT1 (0.64) ALDH1A1HSD17B10HIF1ATSHRHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109311839-B Methylamine derivatives as lysyl oxidase inhibitors for the treatment of cancer 癌症研究协会皇家癌症医院 2021-11-02 CN disclosed
CN-109311839-A Methylamine derivative is used for treating cancer as lysyl oxidase inhibitor 癌症研究协会皇家癌症医院 2019-02-05 CN disclosed