SCHEMBL28657398

SCHEMBL28657398

NC(=O)OCc1ccc(S(=O)(=O)c2ccc(SCCc3ccccc3)cc2)s1

nearest known ligand 0.50

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
LOX P28300 14/20 0.50
CA12 O43570 1/20 0.50
CA1 P00915 1/20 0.50
CA2 P00918 1/20 0.50
CA7 P43166 1/20 0.50
CA13 Q8N1Q1 1/20 0.50
LOXL2 Q9Y4K0 3/20 0.45
MAOA P21397 2/20 0.45
LMNA P02545 1/20 0.41
MCL1 Q07820 4/20 0.39
BCL2A1 Q16548 4/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28652319 0.84 CA2 (0.50) LOXCA12CA1CA2CA7
SCHEMBL19259994 0.81 LOX (0.48) LOXCA12CA1CA2CA7
SCHEMBL28657408 0.79 LOX (0.52) LOXCA2LOXL2MAOA
SCHEMBL28663727 0.78 LOX (0.47) LOXLOXL2MAOA
SCHEMBL19274445 0.77 LOX (0.42) LOXCA12CA1CA2CA7
SCHEMBL31012108 0.77 CA2 (0.75) CA12CA1CA2CA7CA13
SCHEMBL28663650 0.75 LOX (0.57) LOXLOXL2
SCHEMBL28649544 0.75 LOX (0.44) LOXLOXL2MAOALMNA
SCHEMBL28657374 0.75 LOX (0.68) LOXCA2LOXL2
SCHEMBL28643866 0.73 LOX (0.76) LOXLOXL2MAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109311839-B Methylamine derivatives as lysyl oxidase inhibitors for the treatment of cancer 癌症研究协会皇家癌症医院 2021-11-02 CN disclosed