SCHEMBL28658698

SCHEMBL28658698

COC(=O)c1ccccc1Nc1ccc(C)cc1

nearest known ligand 0.78

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.78
ALOX15 P16050 1/20 0.78
SIRT2 Q8IXJ6 2/20 0.61
KDM4E B2RXH2 3/20 0.59
POLB P06746 1/20 0.59
ATM Q13315 1/20 0.59
KMT2A Q03164 3/20 0.55
L3MBTL1 Q9Y468 1/20 0.55
ALDH1A1 P00352 1/20 0.55
ALOX12 P18054 1/20 0.55
PTGS2 P35354 1/20 0.54
NPC1 O15118 1/20 0.53
RAB9A P51151 1/20 0.53
GAA P10253 3/20 0.53
TSHR P16473 1/20 0.53
MAPK1 P28482 1/20 0.53
HSD17B10 Q99714 1/20 0.53
AURKA O14965 1/20 0.52
GLA P06280 1/20 0.51
FFAR4 Q5NUL3 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13224505 0.93 MAPT (0.89) MAPTALOX15SIRT2KDM4EPOLB
SCHEMBL12605599 0.89 MAPT (0.76) MAPTALOX15SIRT2KDM4EPOLB
SCHEMBL12109319 0.88 MAPT (0.81) MAPTALOX15SIRT2KDM4EPOLB
SCHEMBL31914 0.88 MAPT (1.00) MAPTALOX15SIRT2KDM4EPOLB
SCHEMBL28649151 0.85 MAPT (0.81) MAPTALOX15SIRT2KDM4EPOLB
SCHEMBL22452889 0.85 MAPT (0.76) MAPTALOX15SIRT2KDM4EPOLB
SCHEMBL13832955 0.85 MAPT (0.76) MAPTALOX15SIRT2KDM4EPOLB
SCHEMBL22853361 0.85 MAPT (0.76) MAPTALOX15SIRT2KDM4EPOLB
SCHEMBL5993324 0.85 MAPT (0.76) MAPTALOX15SIRT2KDM4EPOLB
SCHEMBL17617073 0.85 MAPT (0.76) MAPTALOX15SIRT2KDM4EPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117043154-A GPCR receptor agonists, pharmaceutical compositions comprising same, and methods of use thereof 卡莫特医疗有限公司 2023-11-10 CN disclosed
CN-113768936-B Application of evodiamine derivative in preparation of medicine for treating superficial fungal infection 南华大学 2023-04-14 CN disclosed
CN-113768936-A Application of evodiamine derivative in preparation of medicine for treating superficial fungal infection 南华大学 2021-12-10 CN disclosed