SCHEMBL28649151

SCHEMBL28649151

COC(=O)c1ccccc1Nc1ccc(-c2ccccc2)cc1

nearest known ligand 0.81

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.81
ALOX15 P16050 1/20 0.81
SIRT2 Q8IXJ6 2/20 0.60
KDM4E B2RXH2 6/20 0.57
POLB P06746 1/20 0.57
ATM Q13315 1/20 0.57
KMT2A Q03164 4/20 0.53
FABP4 P15090 1/20 0.51
CXCR2 P25025 1/20 0.51
AURKA O14965 1/20 0.51
MEN1 O00255 3/20 0.50
SMN1; SMN2 Q16637 2/20 0.50
SIRT1 Q96EB6 1/20 0.50
GLA P06280 1/20 0.50
HTT P42858 1/20 0.50
LMNA P02545 1/20 0.49
PTGS2 P35354 1/20 0.49
SLC6A3 Q01959 1/20 0.49
ALDH1A1 P00352 3/20 0.48
PTGER4 P35408 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12109319 0.97 MAPT (0.81) MAPTALOX15SIRT2KDM4EPOLB
SCHEMBL13224505 0.92 MAPT (0.89) MAPTALOX15SIRT2KDM4EPOLB
SCHEMBL31914 0.90 MAPT (1.00) MAPTALOX15SIRT2KDM4EPOLB
SCHEMBL12109338 0.89 MAPT (0.69) MAPTALOX15SIRT2KDM4EPOLB
SCHEMBL1301699 0.89 MAPT (0.69) MAPTALOX15SIRT2KDM4EPOLB
SCHEMBL22445145 0.86 MAPT (0.79) MAPTALOX15SIRT2KDM4EPOLB
SCHEMBL31168050 0.86 MAPT (0.79) MAPTALOX15SIRT2KDM4EPOLB
SCHEMBL28658698 0.85 MAPT (0.78) MAPTALOX15SIRT2KDM4EPOLB
SCHEMBL27716618 0.84 MAPT (0.67) MAPTALOX15SIRT2KDM4EPOLB
SCHEMBL12605599 0.84 MAPT (0.76) MAPTALOX15SIRT2KDM4EPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115073468-A Preparation and application of imidazopyrazine BTK inhibitor 药雅科技(上海)有限公司 2022-09-20 CN disclosed
CN-113631548-A Serotonin 5-HT2B inhibiting compounds 硕腾服务有限责任公司 2021-11-09 CN disclosed