SCHEMBL28659470

SCHEMBL28659470

F[B-](F)(F)F.F[B-](F)(F)F.F[B-](F)(F)F.Fc1ccc(C[K])cc1

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 5/20 0.46
LOXL2 Q9Y4K0 1/20 0.46
TAAR1 Q96RJ0 3/20 0.42
AGXT P21549 2/20 0.41
PLA2G1B P04054 1/20 0.37
ATG4B Q9Y4P1 1/20 0.37
MAOB P27338 1/20 0.37
MIF P14174 1/20 0.37
LMNA P02545 1/20 0.37
AOC3 Q16853 1/20 0.35
CHRM2 P08172 1/20 0.35
TRPA1 O75762 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31739253 0.76 CALM1 (0.43) IDO1LOXL2TAAR1MAOBTRPA1
SCHEMBL25263956 0.76 CALM1 (0.43) IDO1LOXL2TAAR1MAOBTRPA1
SCHEMBL19260349 0.70 IDO1 (0.48) IDO1LOXL2TAAR1AGXTPLA2G1B
SCHEMBL28314301 0.69 IDO1 (0.39) IDO1LOXL2TAAR1AGXT
Potassium Ion SCHEMBL19260323 0.68 IDO1 (0.46) IDO1LOXL2TAAR1AGXTPLA2G1B
SCHEMBL1468357 0.67 IDO1 (0.58) IDO1LOXL2TAAR1AGXTPLA2G1B
SCHEMBL7437052 0.67 TAAR1 (0.68) IDO1LOXL2TAAR1AGXTMAOB
SCHEMBL16561361 0.67 IDO1 (0.58) IDO1LOXL2TAAR1AGXTPLA2G1B
Lithium Ion SCHEMBL7741416 0.67 IDO1 (0.50) IDO1LOXL2TAAR1AGXTPLA2G1B
SCHEMBL7719447 0.67 IDO1 (0.50) IDO1LOXL2TAAR1AGXTPLA2G1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109071562-B Fused 1, 4-oxazepine and related analogs as BET bromodomain inhibitors 密执安大学评议会 2022-03-22 CN disclosed
CN-110294776-B Method for preparing aryl phosphine oxide derivative 苏州大学 2021-12-10 CN disclosed