SCHEMBL28659989

SCHEMBL28659989

COc1cc(NCc2ccccc2)c(C(=O)O)c(OC)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 1/20 0.56
HDAC8 Q9BY41 3/20 0.53
HDAC1 Q13547 1/20 0.53
HDAC6 Q9UBN7 1/20 0.53
MEN1 O00255 2/20 0.50
KMT2A Q03164 2/20 0.50
L3MBTL1 Q9Y468 2/20 0.50
GAA P10253 1/20 0.50
MAPT P10636 1/20 0.50
CRHBP P24387 1/20 0.50
HTT P42858 1/20 0.50
CRHR2 Q13324 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
APAF1 O14727 1/20 0.48
SENP7 Q9BQF6 1/20 0.48
SENP6 Q9GZR1 1/20 0.48
VNN1 O95497 2/20 0.47
HIF1A Q16665 2/20 0.46
ALDH1A1 P00352 1/20 0.46
MAPK1 P28482 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28655635 0.90 KDM4E (0.46) PTPN1HDAC8HDAC1HDAC6MEN1
SCHEMBL28662381 0.88 L3MBTL1 (0.54) PTPN1MEN1KMT2AL3MBTL1GAA
SCHEMBL28668176 0.88 KMT2A (0.49) PTPN1HDAC8MEN1KMT2AHTT
SCHEMBL28928914 0.84 KMT2A (0.61) MEN1KMT2AL3MBTL1GAAMAPT
SCHEMBL30358562 0.82 CA12 (0.57) HDAC8HDAC1HDAC6MEN1KMT2A
SCHEMBL9956587 0.82 CA12 (0.57) HDAC8HDAC1HDAC6MEN1KMT2A
SCHEMBL31643877 0.80 CYP3A4 (0.51) PTPN1HDAC8HDAC1HDAC6MEN1
SCHEMBL22836927 0.78 AKR1C3 (0.63) L3MBTL1ALDH1A1KDM4EASPHRIOX2
SCHEMBL10787691 0.77 RAB9A (0.55) MEN1KMT2AGAAMAPTSMN1; SMN2
SCHEMBL30691740 0.77 HDAC8 (0.60) HDAC8HDAC1HDAC6MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116270577-A Application of polysubstituted benzene compounds in preparation of medicines for treating cognitive impairment diseases, structure and preparation method 中国医学科学院医药生物技术研究所 2023-06-23 CN disclosed
CN-116270576-A Application of polysubstituted benzene compounds in preparation of medicines for treating cognitive impairment diseases, structure and preparation method 中国医学科学院医药生物技术研究所 2023-06-23 CN disclosed
CN-113521048-B Application of polysubstituted benzene compound in preparation of medicine for treating cognitive disorder diseases, structure and preparation method 中国医学科学院医药生物技术研究所 2023-04-14 CN disclosed
CN-113521048-A Application of polysubstituted benzene compound in preparation of medicine for treating cognitive disorder diseases, structure and preparation method 中国医学科学院医药生物技术研究所 2021-10-22 CN disclosed