SCHEMBL28662969

SCHEMBL28662969

COc1cccc(C(NCc2ccccc2)c2ccccn2)c1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASR P41180 7/20 0.61
DRD2 P14416 1/20 0.50
TDP1 Q9NUW8 1/20 0.46
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
TP53 P04637 2/20 0.44
CYP1A2 P05177 2/20 0.44
CYP3A4 P08684 2/20 0.44
CYP2D6 P10635 2/20 0.44
TSHR P16473 2/20 0.44
MAPK1 P28482 2/20 0.44
CYP2C19 P33261 2/20 0.44
CLK4 Q9HAZ1 2/20 0.44
ALDH1A1 P00352 1/20 0.44
LMNA P02545 1/20 0.44
ALOX15 P16050 1/20 0.44
VDR P11473 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
P4HB P07237 1/20 0.43
MAOB P27338 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28662971 1.00 CASR (0.61) CASRDRD2TDP1MEN1KMT2A
SCHEMBL28928167 0.90 CASR (0.50) CASRDRD2TDP1MEN1KMT2A
SCHEMBL28928166 0.90 CASR (0.50) CASRDRD2TDP1MEN1KMT2A
SCHEMBL28663869 0.86 TDP1 (0.59) CASRTDP1MEN1KMT2ATSHR
SCHEMBL28663870 0.86 TDP1 (0.59) CASRTDP1MEN1KMT2ATSHR
SCHEMBL28669199 0.86 DRD2 (0.46) CASRDRD2ALDH1A1VDRL3MBTL1
SCHEMBL28669200 0.86 DRD2 (0.46) CASRDRD2ALDH1A1VDRL3MBTL1
SCHEMBL28657559 0.83 SLC6A2 (0.50) TDP1MEN1KMT2ACYP1A2ALDH1A1
SCHEMBL28657560 0.83 SLC6A2 (0.50) TDP1MEN1KMT2ACYP1A2ALDH1A1
SCHEMBL28662535 0.81 KDM4E (0.43) ALDH1A1LMNAVDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113683556-B Chiral aryl N-heteroaryl methylamine and preparation method thereof 湖北滋兰生物医药科技有限公司 2024-06-07 CN disclosed
CN-113683556-A Chiral aryl N-heteroaryl methylamine and preparation method thereof 湖北滋兰生物医药科技有限公司 2021-11-23 CN disclosed