SCHEMBL28664347

SCHEMBL28664347

CC(C)(C)OC(=O)c1cccc(-c2cccc(N)n2)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ASIC3 Q9UHC3 1/20 0.46
SLC7A5 Q01650 1/20 0.46
ABCG2 Q9UNQ0 2/20 0.42
ABCB1 P08183 1/20 0.42
LARS1 Q9P2J5 1/20 0.41
CA12 O43570 2/20 0.40
CA1 P00915 2/20 0.40
CA2 P00918 2/20 0.40
CA9 Q16790 2/20 0.40
CA14 Q9ULX7 1/20 0.40
STAT3 P40763 1/20 0.39
PDPK1 O15530 1/20 0.39
SDHB P21912 1/20 0.39
GRM6 O15303 1/20 0.39
IDH1 O75874 1/20 0.38
SCN3A Q9NY46 3/20 0.38
SCN4A P35499 2/20 0.38
GABRG2 P18507 1/20 0.38
GABRB3 P28472 1/20 0.38
GABRA5 P31644 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6714723 0.84 CA12 (0.52) ASIC3LARS1CA12CA1CA2
SCHEMBL28663102 0.83 SLC7A5 (0.43) SLC7A5ABCG2ABCB1CA12CA1
SCHEMBL725997 0.82 SLC7A5 (0.43) SLC7A5ABCG2ABCB1CA12CA1
SCHEMBL31049680 0.82 SLC7A5 (0.43) SLC7A5ABCG2ABCB1CA12CA1
SCHEMBL28669756 0.81 SLC7A5 (0.42) SLC7A5ABCG2ABCB1CA12CA1
SCHEMBL2344130 0.80 SLC7A5 (0.52) SLC7A5CA12CA1CA2CA9
SCHEMBL2031607 0.79 ALDH1A1 (0.41) SLC7A5ABCG2ABCB1CA12CA1
SCHEMBL21056029 0.78 SLC7A5 (0.44) SLC7A5ABCG2ABCB1CA12CA1
SCHEMBL30437476 0.78 SLC7A5 (0.44) SLC7A5ABCG2ABCB1CA12CA1
SCHEMBL31188294 0.78 CA12 (0.49) SLC7A5CA12CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113912617-A Substituted tricycles and methods of use 艾伯维公司 2022-01-11 CN disclosed
CN-108349930-B Substituted tricycles and methods of use 艾伯维公司 2021-10-29 CN disclosed