SCHEMBL28664449

SCHEMBL28664449

CC(NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)NC1(Cc2ccccn2)CCN(C(=O)OC(C)(C)C)CC1

nearest known ligand 0.45

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 1/20 0.45
RET P07949 6/20 0.38
GPR119 Q8TDV5 2/20 0.38
MDM2 Q00987 1/20 0.36
MDM4 O15151 1/20 0.36
TP53 P04637 1/20 0.36
ALOX15 P16050 1/20 0.36
TSHR P16473 1/20 0.36
CNR2 P34972 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29970883 1.00 BACE1 (0.45) BACE1RETGPR119MDM2MDM4
SCHEMBL20137466 0.90 RET (0.39) RETMDM4TP53
SCHEMBL20137467 0.90 RET (0.39) RETMDM4TP53
SCHEMBL20069388 0.84 TLR2 (0.39) RETMDM4TP53
Trifluoroacetic Acid SCHEMBL29971166 0.81 TLR2 (0.38) MDM2MDM4TP53
SCHEMBL28679088 0.79 RET (0.48) RETGPR119ALOX15TSHRCNR2
SCHEMBL29971642 0.79 RET (0.48) RETGPR119ALOX15TSHRCNR2
SCHEMBL2950721 0.77 BACE1 (0.48) BACE1GPR119ALOX15TSHRCNR2
SCHEMBL20069294 0.77 CASP3 (0.45) RET
SCHEMBL20069292 0.77 CASP3 (0.45) RET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110177786-B Substituted pyrazolo [1,5-A ] pyridine compounds as RET kinase inhibitors 阿雷生物药品公司 2021-12-14 CN disclosed