SCHEMBL286658

SCHEMBL286658

Cc1onc(-c2ccc(F)cc2)c1COc1cc(C(=O)NC(C)CO)n(C)n1

nearest known ligand 0.59

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
GABRA5 P31644 20/20 0.59
GABRG2 P18507 1/20 0.48
GABRB3 P28472 1/20 0.48
KCNH2 Q12809 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL286151 1.00 GABRA5 (0.59) GABRA5GABRG2GABRB3KCNH2
SCHEMBL286044 1.00 GABRA5 (0.59) GABRA5GABRG2GABRB3KCNH2
SCHEMBL286291 0.93 GABRA5 (0.68) GABRA5
SCHEMBL2098576 0.90 GABRA5 (0.59) GABRA5
SCHEMBL296065 0.90 GABRA5 (0.59) GABRA5
SCHEMBL297776 0.90 GABRA5 (0.59) GABRA5
SCHEMBL2628064 0.89 GABRA5 (0.60) GABRA5GABRG2GABRB3KCNH2
SCHEMBL285690 0.89 GABRA5 (0.60) GABRA5GABRG2GABRB3KCNH2
SCHEMBL291878 0.86 GABRA5 (0.56) GABRA5
SCHEMBL286356 0.85 GABRA5 (0.54) GABRA5GABRG2GABRB3KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8163728-B2 Pyrazoles HOFFMANN-LA ROCHE INC. (US) 2012-04-24 US disclosed
EP-2427455-A1 ISOXAZOLE-PYRAZOLE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2012-03-14 EP disclosed