SCHEMBL28667748

SCHEMBL28667748

O=C(O)c1cnn2cc(I)cnc12

nearest known ligand 0.47

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.41
ALDH1A1 P00352 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
PDE2A O00408 6/20 0.40
IRAK4 Q9NWZ3 4/20 0.35
POLB P06746 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
HTT P42858 1/20 0.34
HSD11B1 P28845 2/20 0.33
IRAK1 P51617 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19029939 0.82 LMNA (0.47) KDM4EALDH1A1PDE2AIRAK4HSD11B1
SCHEMBL12505413 0.80 IRAK4 (0.43) KDM4EALDH1A1TDP1PDE2AIRAK4
SCHEMBL310362 0.79 HSD11B1 (0.49) KDM4EALDH1A1TDP1PDE2AIRAK4
SCHEMBL310187 0.79 KDM4E (0.43) KDM4EALDH1A1TDP1PDE2AIRAK4
SCHEMBL310126 0.79 PDE2A (0.59) KDM4EALDH1A1TDP1PDE2AHSD11B1
SCHEMBL309283 0.79 KDM4E (0.43) KDM4EALDH1A1TDP1PDE2AIRAK4
SCHEMBL308924 0.77 KDM4E (0.42) KDM4EALDH1A1TDP1PDE2AIRAK4
SCHEMBL12505460 0.76 IRAK4 (0.43) KDM4EALDH1A1TDP1PDE2AIRAK4
SCHEMBL14033080 0.76 KDM4E (0.40) KDM4EALDH1A1TDP1PDE2APOLB
SCHEMBL357836 0.76 LMNA (0.45) KDM4EALDH1A1TDP1PDE2AIRAK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108473498-B Pyrazolo [1,5a ] pyrimidine derivatives as IRAK4 modulators 豪夫迈·罗氏有限公司 2021-11-02 CN disclosed