SCHEMBL28677017

SCHEMBL28677017

COC(=O)c1cccn1CCCCc1ccncc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP4A11 Q02928 3/20 0.43
CYP4F2 P78329 2/20 0.43
HDAC3 O15379 4/20 0.40
HDAC4 P56524 4/20 0.40
HDAC1 Q13547 4/20 0.40
HDAC7 Q8WUI4 4/20 0.40
HDAC2 Q92769 4/20 0.40
HDAC10 Q969S8 4/20 0.40
HDAC11 Q96DB2 4/20 0.40
HDAC8 Q9BY41 4/20 0.40
HDAC6 Q9UBN7 4/20 0.40
HDAC9 Q9UKV0 4/20 0.40
HDAC5 Q9UQL6 4/20 0.40
EP300 Q09472 2/20 0.39
USP2 O75604 1/20 0.39
MAPK10 P53779 1/20 0.39
ALDH1A1 P00352 2/20 0.38
CES1 P23141 2/20 0.38
FLT1 P17948 1/20 0.37
KDR P35968 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24434999 0.96 HDAC3 (0.43) CYP4A11CYP4F2HDAC3HDAC4HDAC1
SCHEMBL24435270 0.91 FLT1 (0.42) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL28677284 0.84 DRD4 (0.43) FLT1KDRDRD4SLC6A4
SCHEMBL24435304 0.84 NPC1 (0.48) CYP4A11CYP4F2HDAC3HDAC4HDAC1
SCHEMBL28677294 0.82 HDAC3 (0.56) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL25395065 0.82 USP2 (0.51) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL24435000 0.80 TBXAS1 (0.45) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL9807560 0.79 CNR1 (0.47) ALDH1A1CNR2
SCHEMBL1422343 0.78 CNR2 (0.47) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL16467932 0.78 CNR2 (0.41) CYP4A11CYP4F2ALDH1A1CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113993587-A Thiazole derivatives as protein secretion inhibitors 科智生命科学公司 2022-01-28 CN disclosed