SCHEMBL28677294

SCHEMBL28677294

COC(=O)c1cccn1CCCc1cccnc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 2/20 0.56
HDAC4 P56524 2/20 0.56
HDAC1 Q13547 2/20 0.56
HDAC7 Q8WUI4 2/20 0.56
HDAC2 Q92769 2/20 0.56
HDAC10 Q969S8 2/20 0.56
HDAC11 Q96DB2 2/20 0.56
HDAC8 Q9BY41 2/20 0.56
HDAC6 Q9UBN7 2/20 0.56
HDAC9 Q9UKV0 2/20 0.56
HDAC5 Q9UQL6 2/20 0.56
KDM4E B2RXH2 2/20 0.47
TBXAS1 P24557 7/20 0.46
TSHR P16473 3/20 0.44
MAPK1 P28482 2/20 0.44
CHRNA7 P36544 1/20 0.44
ALDH1A1 P00352 2/20 0.43
TDP1 Q9NUW8 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
HSP90AA1 P07900 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25394077 0.93 HDAC3 (0.47) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL24434999 0.86 HDAC3 (0.43) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL28681481 0.85 HDAC3 (0.55) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL31466283 0.85 KDM4E (0.57) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL28932117 0.85 KDM4E (0.57) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL24435304 0.84 NPC1 (0.48) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL28677017 0.82 CYP4A11 (0.43) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL28697953 0.80 HDAC3 (0.37) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL24435270 0.78 FLT1 (0.42) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL2333161 0.78 ALDH1A1 (0.56) HDAC1HDAC8KDM4ETSHRMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113993587-A Thiazole derivatives as protein secretion inhibitors 科智生命科学公司 2022-01-28 CN disclosed