SCHEMBL28677352

SCHEMBL28677352

CC(C)(C)OC(=O)NC(CC(=O)O)C(=O)Nc1ccc2[nH]c(C(=O)OC(C)(C)C)cc2c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LEF1 Q9UJU2 1/20 0.49
MMP13 P45452 1/20 0.46
CA12 O43570 1/20 0.45
CA1 P00915 1/20 0.45
CA2 P00918 1/20 0.45
CA4 P22748 1/20 0.45
CA9 Q16790 1/20 0.45
CTNNB1 P35222 9/20 0.44
HDAC4 P56524 2/20 0.43
HDAC1 Q13547 2/20 0.43
SIRT5 Q9NXA8 1/20 0.42
F11 P03951 1/20 0.42
CCKBR P32239 4/20 0.42
HDAC3 O15379 1/20 0.42
HDAC7 Q8WUI4 1/20 0.42
HDAC2 Q92769 1/20 0.42
HDAC10 Q969S8 1/20 0.42
HDAC11 Q96DB2 1/20 0.42
HDAC8 Q9BY41 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28677350 1.00 LEF1 (0.49) LEF1MMP13CA12CA1CA2
SCHEMBL28291191 0.93 MMP13 (0.58) LEF1MMP13CA12CA1CA2
SCHEMBL28291196 0.93 MMP13 (0.58) LEF1MMP13CA12CA1CA2
SCHEMBL23486835 0.92 LEF1 (0.47) LEF1MMP13CTNNB1HDAC4HDAC1
SCHEMBL28681215 0.87 KLK7 (0.46) LEF1MMP13CA12CA1CA2
SCHEMBL28681216 0.87 KLK7 (0.46) LEF1MMP13CA12CA1CA2
SCHEMBL28291195 0.86 CA12 (0.45) LEF1MMP13CA12CA1CA2
SCHEMBL23486833 0.86 LEF1 (0.49) LEF1MMP13CA12CA1CA2
SCHEMBL28692998 0.86 LEF1 (0.44) LEF1MMP13CA12CA1CA2
SCHEMBL28692999 0.86 LEF1 (0.44) LEF1MMP13CA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113943259-A Amino acid derivative, preparation method and application thereof 西安禾渼生物医药有限公司 2022-01-18 CN disclosed