SCHEMBL28677516

SCHEMBL28677516

c1ccc(-c2cc(-c3cccs3)no2)cc1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 8/20 0.65
NPC1 O15118 7/20 0.65
CASP3 P42574 1/20 0.54
SENP8 Q96LD8 1/20 0.54
SENP7 Q9BQF6 1/20 0.54
SENP6 Q9GZR1 1/20 0.54
PTGS2 P35354 2/20 0.48
MEN1 O00255 3/20 0.47
KMT2A Q03164 3/20 0.47
TOP1 P11387 1/20 0.46
ALDH1A1 P00352 3/20 0.46
SMN1; SMN2 Q16637 4/20 0.46
LMNA P02545 1/20 0.46
KDM4E B2RXH2 2/20 0.45
MAPT P10636 2/20 0.45
CYP1A2 P05177 2/20 0.45
HPGD P15428 2/20 0.45
CYP2C9 P11712 1/20 0.45
NFKB1 P19838 1/20 0.45
CYP2C19 P33261 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28677256 0.86 NPC1 (0.65) RAB9ANPC1CASP3SENP8SENP7
3,5-Diphenylisoxazole SCHEMBL1421260 0.79 NPC1 (1.00) RAB9ANPC1CASP3SENP8SENP7
SCHEMBL8258186 0.77 NPC1 (0.96) RAB9ANPC1CASP3SENP8SENP7
SCHEMBL7211172 0.75 CYP1A2 (0.41) RAB9AMEN1KMT2AALDH1A1SMN1; SMN2
SCHEMBL14896296 0.75 HSD17B10 (0.50) RAB9ANPC1CASP3SENP8SENP7
SCHEMBL11961408 0.75 ALDH1A1 (0.50) RAB9ANPC1CASP3SENP8SENP7
SCHEMBL7020024 0.75 KDM4E (0.47) RAB9ANPC1CASP3SENP8SENP7
SCHEMBL5904743 0.75 KDM4E (0.47) RAB9ANPC1CASP3SENP8SENP7
SCHEMBL27847623 0.74 KDM4E (0.46) RAB9ANPC1CASP3SENP8SENP7
SCHEMBL17874000 0.73 KDM4E (0.47) RAB9ANPC1MEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113248455-A 3, 5-disubstituted isoxazole derivatives and synthesis method thereof 湖北科技学院 2021-08-13 CN disclosed