SCHEMBL28677772

SCHEMBL28677772

CC(=O)OC(C)(N1Cc2ccccc2C1)C(F)(F)F

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 3/20 0.43
MAPT P10636 2/20 0.43
TAAR1 Q96RJ0 2/20 0.43
LMNA P02545 1/20 0.43
HSP90AA1 P07900 1/20 0.39
HSD17B3 P37058 3/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
RIPK1 Q13546 2/20 0.37
ABHD6 Q9BV23 1/20 0.37
NAMPT P43490 2/20 0.35
MAPK1 P28482 1/20 0.35
PDK1 Q15118 2/20 0.34
PDK2 Q15119 2/20 0.34
PDK3 Q15120 2/20 0.34
PDK4 Q16654 2/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL31197675 0.71 NOTUM (0.42) NOTUMMAPTTAAR1LMNAHSP90AA1
SCHEMBL31292095 0.69 NOTUM (0.50) NOTUMHSP90AA1HSD17B3NPC1RAB9A
SCHEMBL31292601 0.68 NOTUM (0.46) NOTUMMAPTTAAR1LMNAHSP90AA1
SCHEMBL861946 0.65 MAOA (0.44) NOTUMMAPTHSD17B3NPC1RAB9A
SCHEMBL29676965 0.65 MAPK1 (0.64) NOTUMRIPK1NAMPTMAPK1
SCHEMBL21947725 0.65 CYP2C19 (0.44) MAPTLMNAMAPK1PDK1PDK2
SCHEMBL5183098 0.65 MAPK1 (0.64) NOTUMRIPK1NAMPTMAPK1
SCHEMBL6204851 0.65 MAPK1 (0.52) NOTUMRIPK1NAMPTMAPK1MEN1
SCHEMBL27570729 0.64 CYP2C19 (0.47) MAPTMAPK1PDK1PDK2PDK3
SCHEMBL20609569 0.63 ALDH1A1 (0.42) NOTUMMAPTTAAR1LMNAHSP90AA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113993591-A Novel EGFR inhibitors 豪夫迈·罗氏有限公司 2022-01-28 CN disclosed
CN-113993590-A Novel EGFR inhibitors 豪夫迈·罗氏有限公司 2022-01-28 CN disclosed