SCHEMBL28677828

SCHEMBL28677828

CCn1c(=O)c(C(=O)O)c(O)c2cc(Cl)ccc21

nearest known ligand 0.75

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.75
GSK3B P49841 4/20 0.62
MEN1 O00255 5/20 0.56
KMT2A Q03164 5/20 0.56
PTGER4 P35408 1/20 0.51
KDM4E B2RXH2 4/20 0.50
HTT P42858 2/20 0.50
LMNA P02545 2/20 0.50
POLB P06746 1/20 0.50
TDP1 Q9NUW8 1/20 0.50
MAPT P10636 1/20 0.47
HPGD P15428 1/20 0.47
MAPK1 P28482 1/20 0.47
HSD17B10 Q99714 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28515304 0.89 GSK3B (0.62) ALDH1A1GSK3BMEN1KMT2AKDM4E
SCHEMBL15966835 0.86 ALDH1A1 (1.00) ALDH1A1GSK3BMEN1KMT2AKDM4E
SCHEMBL28519313 0.84 ALDH1A1 (0.58) ALDH1A1GSK3BMEN1KMT2AKDM4E
SCHEMBL28511432 0.83 ALDH1A1 (0.54) ALDH1A1GSK3BMEN1KMT2AKDM4E
SCHEMBL11372872 0.83 GSK3B (0.57) ALDH1A1GSK3BMEN1KMT2A
SCHEMBL28511846 0.81 KDM4E (0.68) ALDH1A1MEN1KMT2APTGER4KDM4E
SCHEMBL7435419 0.80 KDM4E (0.72) ALDH1A1MEN1KMT2AKDM4EHTT
SCHEMBL28678706 0.79 KMT2A (0.55) ALDH1A1GSK3BMEN1KMT2AKDM4E
SCHEMBL11379590 0.78 GSK3B (0.60) GSK3BMEN1KMT2AKDM4ELMNA
SCHEMBL15966782 0.78 GSK3B (1.00) GSK3BMEN1KMT2AKDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110041306-B 4-hydroxy-2-quinolone-N- (4-quinazolinone) -3-carboxamide derivatives 中国医学科学院药物研究所 2022-01-11 CN disclosed