SCHEMBL28680245

SCHEMBL28680245

COC(=O)c1cccc(-c2nc(Br)c[nH]2)c1

nearest known ligand 0.54

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CDK8 P49336 1/20 0.54
NEK1 Q96PY6 5/20 0.50
AXL P30530 1/20 0.50
ASH1L Q9NR48 1/20 0.46
GABRG2 P18507 1/20 0.46
GABRB3 P28472 1/20 0.46
GABRA5 P31644 1/20 0.46
GABRA3 P34903 1/20 0.46
CA12 O43570 1/20 0.46
CA1 P00915 1/20 0.46
CA2 P00918 1/20 0.46
CA9 Q16790 1/20 0.46
PLAU P00749 3/20 0.46
ERN1 O75460 2/20 0.45
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
SDHB P21912 1/20 0.44
LOXL2 Q9Y4K0 1/20 0.42
NPY5R Q15761 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27949967 0.84 CDK8 (0.55) CDK8NEK1AXLASH1LGABRG2
SCHEMBL7461576 0.84 CDK8 (0.55) CDK8NEK1AXLASH1LGABRG2
SCHEMBL17279808 0.84 CDK8 (0.55) CDK8NEK1AXLASH1LGABRG2
SCHEMBL30107993 0.81 CDK8 (0.54) CDK8NEK1AXLGABRG2GABRB3
SCHEMBL29215207 0.79 CDK8 (0.50) CDK8NEK1AXLGABRG2GABRB3
SCHEMBL67941 0.77 CA12 (0.68) CDK8GABRG2GABRB3GABRA5GABRA3
SCHEMBL5184668 0.76 CDK8 (0.47) CDK8NEK1AXLASH1LGABRG2
SCHEMBL28871291 0.76 PKN1 (0.52) CDK8GABRG2GABRB3GABRA5GABRA3
SCHEMBL3062520 0.75 KDM4E (0.70) CDK8NEK1AXLASH1LGABRG2
SCHEMBL17280197 0.75 ALDH1A1 (0.54) CDK8NEK1AXLPLAUNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113767105-A Heterocyclic compounds as inhibitors of monoacylglycerol lipases (MAGL) 豪夫迈·罗氏有限公司 2021-12-07 CN disclosed