SCHEMBL30107993

SCHEMBL30107993

COC(=O)c1cccc(-c2cccc(Br)n2)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK8 P49336 1/20 0.54
GABRG2 P18507 1/20 0.52
GABRB3 P28472 1/20 0.52
GABRA5 P31644 1/20 0.52
GABRA3 P34903 1/20 0.52
SDHB P21912 1/20 0.49
CA12 O43570 1/20 0.49
CA1 P00915 1/20 0.49
CA2 P00918 1/20 0.49
CA9 Q16790 1/20 0.49
PLAU P00749 4/20 0.48
ABL1 P00519 1/20 0.48
BCR P11274 1/20 0.48
SRC P12931 1/20 0.48
ERN1 O75460 2/20 0.48
NEK1 Q96PY6 2/20 0.47
NPC1 O15118 1/20 0.47
RAB9A P51151 1/20 0.47
AXL P30530 1/20 0.47
KDM5B Q9UGL1 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6718372 0.85 CNR1 (0.56) CDK8GABRG2GABRB3GABRA5GABRA3
SCHEMBL4895475 0.84 GABRG2 (0.66) CDK8GABRG2GABRB3GABRA5GABRA3
SCHEMBL4901644 0.84 TP53 (0.50) NPC1RAB9A
SCHEMBL13680584 0.83 GABRG2 (0.53) CDK8GABRG2GABRB3GABRA5GABRA3
SCHEMBL6714723 0.82 CA12 (0.52) CDK8GABRG2GABRB3GABRA5GABRA3
SCHEMBL28680245 0.81 CDK8 (0.54) CDK8GABRG2GABRB3GABRA5GABRA3
SCHEMBL16553302 0.80 GABRG2 (0.53) CDK8GABRG2GABRB3GABRA5GABRA3
SCHEMBL67941 0.80 CA12 (0.68) CDK8GABRG2GABRB3GABRA5GABRA3
SCHEMBL21790698 0.79 GABRG2 (0.50) CDK8GABRG2GABRB3GABRA5GABRA3
SCHEMBL6717982 0.79 CNR1 (0.55) CDK8GABRG2GABRB3GABRA5GABRA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022203399-A1 ADENOSINE A2A RECEPTOR ANTAGONIST AND USE THEREOF 주식회사 스탠다임 2022-09-29 WO disclosed