SCHEMBL28680795

SCHEMBL28680795

OCc1nc2c(Cl)cccc2s1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 4/20 0.56
PDE10A Q9Y233 1/20 0.56
MAPT P10636 4/20 0.51
GAA P10253 2/20 0.51
HPGD P15428 2/20 0.51
KMT2A Q03164 2/20 0.51
ALDH1A1 P00352 2/20 0.51
MAPK1 P28482 2/20 0.51
MEN1 O00255 1/20 0.51
PKM P14618 1/20 0.51
TDP1 Q9NUW8 1/20 0.51
PSMB8 P28062 1/20 0.51
RAB9A P51151 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
AKR1B1 P15121 1/20 0.45
DRD2 P14416 1/20 0.43
DRD4 P21917 1/20 0.43
DRD3 P35462 1/20 0.43
NPC1 O15118 1/20 0.43
NPSR1 Q6W5P4 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30513858 1.00 LMNA (0.56) LMNAPDE10AMAPTGAAHPGD
SCHEMBL23478496 0.82 LMNA (0.61) LMNAPDE10AMAPTGAAHPGD
SCHEMBL7457013 0.82 LMNA (0.56) LMNAPDE10AMAPTGAAHPGD
SCHEMBL6630437 0.82 LMNA (0.56) LMNAPDE10AMAPTGAAHPGD
SCHEMBL24287678 0.80 PDPK1 (0.58) LMNAMAPTGAAHPGDKMT2A
SCHEMBL16674780 0.79 GAA (0.51) LMNAPDE10AMAPTGAAHPGD
SCHEMBL28478793 0.79 SMN1; SMN2 (0.56) LMNAMAPTGAAHPGDKMT2A
SCHEMBL29691142 0.78 DRD2 (0.55) LMNAPDE10AMAPTGAAHPGD
SCHEMBL16806283 0.78 LMNA (0.51) LMNAPDE10AMAPTGAAHPGD
SCHEMBL9037145 0.78 PSMB8 (0.59) LMNAPDE10AMAPTGAAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113816948-B Condensed imidazole derivative, preparation method and medical application thereof 江苏恒瑞医药股份有限公司 2023-08-11 CN disclosed
CN-113816948-A Condensed imidazole derivative, preparation method and application thereof in medicine 江苏恒瑞医药股份有限公司 2021-12-21 CN disclosed