SCHEMBL28684152

SCHEMBL28684152

NC(CCCCC1CNCCO1)CCCN1C(=O)c2cccc3c(-c4ccn[nH]4)ccc1c23

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1B1 Q16678 2/20 0.33
KDM4E B2RXH2 2/20 0.32
SLC6A2 P23975 9/20 0.32
SLC6A4 P31645 9/20 0.32
SLC6A3 Q01959 5/20 0.32
HTR1A P08908 2/20 0.31
DRD2 P14416 2/20 0.31
HTR2A P28223 2/20 0.31
HTR7 P34969 2/20 0.31
HTR6 P50406 2/20 0.31
ALDH1A1 P00352 2/20 0.30
MAPT P10636 2/20 0.30
APAF1 O14727 1/20 0.30
GAA P10253 1/20 0.30
THRB P10828 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30
MEN1 O00255 1/20 0.30
NPC1 O15118 1/20 0.30
S1PR4 O95977 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28696297 0.81 HEXA (0.41) CYP1B1KDM4EHTR1ADRD2HTR2A
SCHEMBL28684148 0.81 KDM4E (0.44) KDM4EHTR1ADRD2HTR2AHTR7
SCHEMBL28689910 0.80 HTR1A (0.44) HTR1ADRD2HTR2AHTR7HTR6
SCHEMBL28695945 0.79 HTR1A (0.43) HTR1ADRD2HTR2AHTR7HTR6
SCHEMBL28703527 0.78 BCHE (0.38) CYP1B1KDM4EALDH1A1MAPTAPAF1
SCHEMBL8555421 0.69 SLC6A2 (0.47) KDM4ESLC6A2SLC6A4SLC6A3HTR1A
SCHEMBL8559698 0.68 TDP1 (0.48) KDM4ESLC6A2SLC6A4SLC6A3HTR1A
SCHEMBL8559794 0.68 TDP1 (0.48) KDM4ESLC6A2SLC6A4SLC6A3HTR1A
SCHEMBL8559087 0.68 TDP1 (0.48) KDM4ESLC6A2SLC6A4SLC6A3HTR1A
SCHEMBL8558048 0.68 TDP1 (0.48) KDM4ESLC6A2SLC6A4SLC6A3HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109665987-B Naphthaleneimide-polyamine conjugates, methods of making and uses thereof 河南大学 2022-02-18 CN disclosed