SCHEMBL28684148

SCHEMBL28684148

NC(CCCCN1CCOCC1)CCCN1C(=O)c2cccc3c(-c4ccn[nH]4)ccc1c23

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.44
MEN1 O00255 1/20 0.44
ALDH1A1 P00352 1/20 0.44
CASP1 P29466 1/20 0.44
CASP7 P55210 1/20 0.44
KMT2A Q03164 1/20 0.44
HSD17B10 Q99714 1/20 0.44
HTR1A P08908 11/20 0.44
HTR7 P34969 10/20 0.44
DRD2 P14416 10/20 0.44
HTR6 P50406 10/20 0.44
HTR2A P28223 9/20 0.44
RORC P51449 1/20 0.42
HDAC3 O15379 2/20 0.41
HDAC1 Q13547 2/20 0.41
HDAC11 Q96DB2 2/20 0.41
NCOR2 Q9Y618 2/20 0.41
HDAC2 Q92769 1/20 0.41
HDAC8 Q9BY41 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28689910 0.92 HTR1A (0.44) HTR1AHTR7DRD2HTR6HTR2A
SCHEMBL28695945 0.92 HTR1A (0.43) MEN1KMT2AHTR1AHTR7DRD2
SCHEMBL28696297 0.85 HEXA (0.41) KDM4EALDH1A1HTR1AHTR7DRD2
SCHEMBL28693048 0.83 HTR7 (0.44) KDM4EMEN1ALDH1A1CASP1CASP7
SCHEMBL28703527 0.81 BCHE (0.38) KDM4EMEN1ALDH1A1KMT2A
SCHEMBL28684152 0.81 CYP1B1 (0.33) KDM4EMEN1ALDH1A1KMT2AHTR1A
SCHEMBL28296691 0.74 PARP1 (0.40) HTR7PARP1
SCHEMBL28704987 0.67 HEXA (0.41) KDM4EMEN1ALDH1A1CASP1CASP7
SCHEMBL28684142 0.67 PDE10A (0.43) KDM4EALDH1A1HSD17B10HTR1AHTR7
SCHEMBL28704128 0.66 CYP1B1 (0.60) KDM4EMEN1ALDH1A1KMT2AHTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109665987-B Naphthaleneimide-polyamine conjugates, methods of making and uses thereof 河南大学 2022-02-18 CN disclosed