SCHEMBL28684653

SCHEMBL28684653

CC(C)(C)OC(=O)NC(CCCNc1ccccc1[N+](=O)[O-])C(=O)O

nearest known ligand 0.49

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.49
TSHR P16473 1/20 0.49
BCL2 P10415 2/20 0.48
KAT2B Q92831 2/20 0.47
PPARA Q07869 3/20 0.45
PPARG P37231 2/20 0.45
CTSK P43235 4/20 0.45
NPC1 O15118 1/20 0.45
MAPT P10636 1/20 0.45
RAB9A P51151 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
DGAT1 O75907 1/20 0.44
JAK3 P52333 1/20 0.44
BTK Q06187 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28684650 1.00 ALDH1A1 (0.49) ALDH1A1TSHRBCL2KAT2BPPARA
SCHEMBL28684687 0.91 GSTP1 (0.48) ALDH1A1TSHRBCL2KAT2BCTSK
SCHEMBL28684688 0.91 GSTP1 (0.48) ALDH1A1TSHRBCL2KAT2BCTSK
SCHEMBL645782 0.87 PPARA (0.48) ALDH1A1TSHRBCL2PPARAPPARG
SCHEMBL949969 0.87 PPARA (0.48) ALDH1A1TSHRBCL2PPARAPPARG
SCHEMBL4704052 0.87 PPARA (0.48) ALDH1A1TSHRBCL2PPARAPPARG
SCHEMBL9300334 0.87 KAT2B (0.51) ALDH1A1TSHRBCL2KAT2BPPARA
SCHEMBL28698446 0.85 KAT2B (0.47) ALDH1A1BCL2KAT2BNPC1MAPT
SCHEMBL29465810 0.85 KAT2B (0.47) ALDH1A1BCL2KAT2BNPC1MAPT
SCHEMBL30849526 0.81 ALDH1A1 (0.61) ALDH1A1KAT2BNPC1MAPTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114057771-B Macrocyclic compounds, their preparation and use 北京鞍石生物科技有限责任公司 2023-10-03 CN disclosed
CN-114057771-A Macrocyclic compound and preparation method and application thereof 北京鞍石生物科技有限责任公司 2022-02-18 CN disclosed