SCHEMBL9300334

SCHEMBL9300334

Cc1ccc([N+](=O)[O-])c(NCCC[C@@H](NC(=O)OC(C)(C)C)C(=O)O)c1

nearest known ligand 0.63

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KAT2B Q92831 3/20 0.51
ALDH1A1 P00352 1/20 0.49
TSHR P16473 1/20 0.49
BCL2 P10415 2/20 0.43
PPARG P37231 2/20 0.43
PPARA Q07869 2/20 0.43
GUCY1A1 Q02108 1/20 0.41
GUCY1B1 Q02153 1/20 0.41
FOLH1 Q04609 2/20 0.41
GSTP1 P09211 1/20 0.41
GSTM2 P28161 1/20 0.41
MAPT P10636 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9387675 0.90 KAT2B (0.47) KAT2BALDH1A1TSHRBCL2PPARG
SCHEMBL28684653 0.87 ALDH1A1 (0.49) KAT2BALDH1A1TSHRBCL2PPARG
SCHEMBL28684650 0.87 ALDH1A1 (0.49) KAT2BALDH1A1TSHRBCL2PPARG
SCHEMBL9391766 0.86 KAT2B (0.51) KAT2BALDH1A1BCL2GSTP1GSTM2
SCHEMBL9391236 0.86 KAT2B (0.57) KAT2BALDH1A1FOLH1MAPT
SCHEMBL9386630 0.85 KAT2B (0.50) KAT2BALDH1A1MAPT
SCHEMBL9388577 0.84 KAT2B (0.53) KAT2BALDH1A1FOLH1MAPT
SCHEMBL9387741 0.83 KAT2B (0.46) KAT2BALDH1A1TSHRBCL2MAPT
SCHEMBL9386631 0.83 KAT2B (0.46) KAT2BALDH1A1TSHRBCL2MAPT
SCHEMBL14981761 0.82 KAT2B (0.58) KAT2BALDH1A1TSHRGUCY1A1GUCY1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1994012163-A1 2-NITROARYL AND 2-CYANOARYL COMPOUNDS AS REGULATORS OF NITRIC OXIDE SYNTHASE ABBOTT LABORATORIES (US) 1994-06-09 WO claimed
US-5362747-A Promoters, inhibitors ABBOTT LABORATORIES (US) 1994-11-08 US disclosed
WO-1994012163-A1 2-NITROARYL AND 2-CYANOARYL COMPOUNDS AS REGULATORS OF NITRIC OXIDE SYNTHASE ABBOTT LABORATORIES (US) 1994-06-09 WO disclosed