SCHEMBL28684668

SCHEMBL28684668

COc1ccc(NC(=O)C(C)(C)C)cc1C

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.56
CYP2C9 P11712 1/20 0.56
CYP2C19 P33261 1/20 0.56
L3MBTL1 Q9Y468 1/20 0.56
LMNA P02545 2/20 0.53
MAPT P10636 2/20 0.50
IMPDH2 P12268 1/20 0.50
IMPDH1 P20839 1/20 0.50
IDO1 P14902 1/20 0.48
TDO2 P48775 1/20 0.48
NPSR1 Q6W5P4 1/20 0.47
LCK P06239 1/20 0.47
CTSL P07711 1/20 0.47
PTPRC P08575 1/20 0.47
PTPN2 P17706 1/20 0.47
PTPN1 P18031 1/20 0.47
CTSS P25774 1/20 0.47
PTPN13 Q12923 1/20 0.47
CYP3A4 P08684 1/20 0.46
ALDH1A1 P00352 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9447193 0.87 CYP1A2 (0.56) CYP1A2CYP2C9CYP2C19L3MBTL1LMNA
SCHEMBL8102792 0.87 CYP1A2 (0.73) CYP1A2CYP2C9CYP2C19L3MBTL1LMNA
SCHEMBL5952099 0.81 ALDH1A1 (0.62) LMNAMAPTALDH1A1KDM4E
SCHEMBL18467344 0.81 ALDH1A1 (0.58) CYP1A2CYP2C9CYP2C19IMPDH2IMPDH1
SCHEMBL14667344 0.81 L3MBTL1 (0.67) CYP1A2L3MBTL1MAPTNPSR1LCK
SCHEMBL5404961 0.80 CYP2C9 (0.60) CYP1A2CYP2C9CYP2C19L3MBTL1LMNA
SCHEMBL14496900 0.80 MAPT (0.53) CYP1A2CYP2C9CYP2C19L3MBTL1LMNA
SCHEMBL1285002 0.79 CYP1A2 (0.59) CYP1A2CYP2C9CYP2C19L3MBTL1LMNA
SCHEMBL30223469 0.79 CYP1A2 (0.59) CYP1A2CYP2C9CYP2C19L3MBTL1LMNA
SCHEMBL344338 0.79 GRM4 (0.57) CYP1A2CYP2C9CYP2C19L3MBTL1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113912529-B Method for synthesizing indole compounds by catalyzing N-aryl amide compounds and vinylene carbonate with ruthenium 成都大学 2023-07-25 CN disclosed
CN-113912529-A Method for synthesizing indole compound by catalyzing N-aryl amide compound and vinylene carbonate with ruthenium 成都大学 2022-01-11 CN disclosed