SCHEMBL28686197

SCHEMBL28686197

COc1ccc(CN(C)c2cnc(-c3ccccc3)c(-c3ccccc3)n2)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CKS1B P61024 2/20 0.55
SKP1 P63208 2/20 0.55
SKP2 Q13309 2/20 0.55
ALDH1A1 P00352 3/20 0.48
LMNA P02545 3/20 0.48
TDP1 Q9NUW8 2/20 0.48
KDM4E B2RXH2 1/20 0.48
NPSR1 Q6W5P4 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
CYP19A1 P11511 1/20 0.44
CNR1 P21554 2/20 0.44
TSHR P16473 3/20 0.43
KMT2A Q03164 2/20 0.43
MEN1 O00255 1/20 0.43
CYP1A2 P05177 1/20 0.43
CHRM2 P08172 1/20 0.43
CYP3A4 P08684 1/20 0.43
HTR1A P08908 1/20 0.43
ADRA2A P08913 1/20 0.43
CYP2D6 P10635 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30725777 1.00 CKS1B (0.55) CKS1BSKP1SKP2ALDH1A1LMNA
SCHEMBL16451103 0.86 CKS1B (0.51) CKS1BSKP1SKP2ALDH1A1LMNA
SCHEMBL30725791 0.85 CKS1B (0.59) CKS1BSKP1SKP2ALDH1A1LMNA
SCHEMBL28690986 0.85 CKS1B (0.59) CKS1BSKP1SKP2ALDH1A1LMNA
SCHEMBL28691774 0.84 CKS1B (0.57) CKS1BSKP1SKP2LMNAKDM4E
SCHEMBL30725778 0.84 CKS1B (0.57) CKS1BSKP1SKP2LMNAKDM4E
SCHEMBL30725764 0.84 CKS1B (0.57) CKS1BSKP1SKP2ALDH1A1LMNA
SCHEMBL28691799 0.84 CKS1B (0.57) CKS1BSKP1SKP2ALDH1A1LMNA
SCHEMBL28697301 0.82 CKS1B (0.55) CKS1BSKP1SKP2LMNANPSR1
SCHEMBL30725783 0.82 CNR1 (0.62) CKS1BSKP1SKP2ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118206499-A 2,3, 5-Trisubstituted pyrazine compound and preparation method and application thereof 郑州大学 2024-06-18 CN disclosed
CN-118146165-A 2,3, 5-Trisubstituted pyrazine compound and preparation method and application thereof 郑州大学 2024-06-07 CN disclosed
CN-113968824-B 2,3, 5-trisubstituted pyrazine compound and preparation method and application thereof 郑州大学 2024-01-19 CN disclosed
CN-113968824-A 2,3, 5-trisubstituted pyrazine compound and preparation method and application thereof 郑州大学 2022-01-25 CN disclosed