SCHEMBL28689290

SCHEMBL28689290

C#CC(OC(C#C)c1ccc(Br)cc1)c1ccc(Br)cc1

nearest known ligand 0.39

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PYCR1 P32322 4/20 0.39
CYP2A6 P11509 1/20 0.36
HTR2A P28223 1/20 0.33
CYP1A2 P05177 1/20 0.32
ESR1 P03372 1/20 0.32
ESR2 Q92731 1/20 0.32
POLB P06746 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28704077 0.77 IDO1 (0.40) CYP2A6ESR1ESR2
SCHEMBL28678690 0.77 IDO1 (0.41) ESR1ESR2
SCHEMBL8408252 0.77 MEN1 (0.36) ESR1ESR2
SCHEMBL77245 0.76 DPP4 (0.36) HTR2ACYP1A2
SCHEMBL28865706 0.75 PYCR1 (0.36) PYCR1HTR2ACYP1A2
SCHEMBL28865707 0.75 PYCR1 (0.36) PYCR1HTR2ACYP1A2
SCHEMBL9834505 0.74 CA1 (0.46) CYP1A2
SCHEMBL28699231 0.74 CYP19A1 (0.40) CYP2A6
SCHEMBL28684586 0.72 PDE2A (0.41) PYCR1
SCHEMBL23244675 0.70 PYCR1 (0.40) PYCR1CYP2A6HTR2ACYP1A2ESR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109336829-B Aryl formamide compound containing 1,2, 3-triazole structure and application thereof 沈阳药科大学 2022-03-01 CN disclosed