SCHEMBL28699510

SCHEMBL28699510

COc1cc(-c2c3c(nn2-c2ccccc2)CCCC3)cc(OC)c1OC

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 1/20 0.50
PDE4B Q07343 1/20 0.50
PDE4C Q08493 1/20 0.50
PDE4D Q08499 1/20 0.50
HTR2A P28223 1/20 0.48
HTR2C P28335 1/20 0.48
HTR2B P41595 1/20 0.48
MAPT P10636 3/20 0.47
NPC1 O15118 1/20 0.45
BCHE P06276 3/20 0.43
ACHE P22303 2/20 0.43
PTGS1 P23219 1/20 0.43
PTGS2 P35354 1/20 0.43
MEN1 O00255 3/20 0.42
KMT2A Q03164 3/20 0.42
LMNA P02545 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28705568 0.99 PDE4A (0.49) PDE4APDE4BPDE4CPDE4DHTR2A
SCHEMBL28261225 0.89 PTGS2 (0.45) PDE4APDE4BPDE4CPDE4DMAPT
SCHEMBL28709337 0.88 PTGS2 (0.45) PDE4APDE4BPDE4CPDE4DMAPT
SCHEMBL29374174 0.88 PDE4A (0.61) PDE4APDE4BPDE4CPDE4DHTR2A
SCHEMBL28700876 0.88 PDE4A (0.61) PDE4APDE4BPDE4CPDE4DHTR2A
SCHEMBL29374838 0.88 TUBB4A (0.43) PDE4APDE4BPDE4CPDE4DHTR2A
SCHEMBL28705573 0.88 TUBB4A (0.43) PDE4APDE4BPDE4CPDE4DHTR2A
SCHEMBL28691204 0.87 PTGS2 (0.45) NPC1PTGS1PTGS2KDM4EMAPK1
SCHEMBL28709340 0.87 BCHE (0.43) PDE4APDE4BPDE4CPDE4DBCHE
SCHEMBL21157448 0.79 HTR2A (0.68) HTR2AHTR2CHTR2BPTGS1PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109020890-B Preparation and application of saturated aliphatic cyclo-pyrazole derivatives 南京大学 2022-02-08 CN disclosed