SCHEMBL28699525

SCHEMBL28699525

O=C(Oc1cc(CN2CCNCC2)cc(C(F)(F)F)c1)C1CC1

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 5/20 0.47
CYP2D6 P10635 4/20 0.47
TSHR P16473 3/20 0.43
CHRM3 P20309 2/20 0.41
USP2 O75604 5/20 0.41
CYP2C19 P33261 3/20 0.41
CYP1A2 P05177 2/20 0.41
MEN1 O00255 1/20 0.41
TP53 P04637 1/20 0.41
KMT2A Q03164 1/20 0.41
MGLL Q99685 2/20 0.41
DDR1 Q08345 1/20 0.41
ALDH1A1 P00352 1/20 0.40
HPGD P15428 1/20 0.38
BRAF P15056 1/20 0.38
KDR P35968 1/20 0.38
CYP2C9 P11712 2/20 0.38
SIGMAR1 Q99720 2/20 0.38
HIF1A Q16665 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29170862 0.96 CYP2D6 (0.46) CYP3A4CYP2D6TSHRCHRM3USP2
SCHEMBL28322502 0.83 CYP2D6 (0.48) CYP3A4CYP2D6TSHRCHRM3USP2
SCHEMBL28936361 0.81 MGLL (0.47) CYP3A4CYP2D6TSHRUSP2CYP2C19
SCHEMBL28705661 0.80 MGLL (0.65) CYP2D6MGLL
SCHEMBL20179998 0.78 CYP3A4 (0.56) CYP3A4CYP2D6TSHRUSP2CYP2C19
SCHEMBL19262510 0.77 CYP2D6 (0.72) CYP3A4CYP2D6TSHRCHRM3USP2
SCHEMBL27586950 0.77 KMT2A (0.47) MEN1KMT2A
SCHEMBL29560940 0.76 CYP2D6 (0.52) CYP3A4CYP2D6TSHRCHRM3USP2
SCHEMBL20137096 0.76 CYP2D6 (0.52) CYP3A4CYP2D6TSHRCHRM3USP2
SCHEMBL20676125 0.76 CYP2D6 (0.70) CYP3A4CYP2D6TSHRCHRM3USP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110267963-B MAGL inhibitors H.隆德贝克有限公司 2022-04-01 CN disclosed